Androgen Receptors

More Information »Androgen receptors (ARs) (dihydrotestosterone receptors) are nuclear hormone receptors of the NR3C class, which includes mineralocorticoid, progesterone and glucocorticoid receptors. ARs are expressed in bone marrow, mammary gland and prostate tissues.

Androgen Receptor Products

Agonists
Cat.No.	Product Name / Activity
3812	Cl-4AS-1
	Steroidal androgen receptor agonist
2822	Testosterone
	Endogenous androgen receptor agonist
Antagonists
Cat.No.	Product Name / Activity
3389	Bicalutamide
	Non-steroidal androgen receptor antagonist
4094	Flutamide
	Non-steroidal androgen receptor antagonist
1759	Nilutamide
	Androgen receptor antagonist. Orally active
3923	PF 998425
	Non-steroidal androgen receptor antagonist
Modulators
Cat.No.	Product Name / Activity
3813	TFM-4AS-1
	Selective androgen receptor modulator (SARM)
Other
Cat.No.	Product Name / Activity
4626	Andrographolide
	Inhibits NFκB; blocks androgen receptor (AR) expression
3293	Finasteride
	Type II 5α-reductase inhibitor
3572	GSK 650394
	Serum- and glucocorticoid-regulated kinase (SGK) inhibitor
4396	Piperlongumine
	Induces apoptosis; depletes androgen receptors in prostate cancer cells
2968	Spironolactone
	Antiandrogen; inhibits steroid hormone biosynthesis. Also MR antagonist