R&D Systems Inc. Tocris Bioscience Boston Biochem

TRPV

More Information »Vanilloids are a group of compounds, structurally related to capsaicin, thought to exert their actions via vanilloid receptors. The vanilloid receptor family (TRPV) is a member of the transient receptor potential (TRP) superfamily of ion channels, and have six members (TRPV1-6).

TRPV Products

Agonists
Cat.No.
Product Name / Activity
1116 AM 404
Vanilloid receptor agonist. Also anandamide transport inhibitor
1685 AM 404 (in Tocrisolve™ 100)
Vanilloid receptor agonist. Also anandamide transport inhibitor (in water-soluble emulsion)
1339 Anandamide
Endogenous CB and TRPV1 receptor agonist
1017 Anandamide (in Tocrisolve™ 100)
Endogenous CB and TRPV1 receptor agonist (in water-soluble emulsion)
1354 Arvanil
Potent TRPV1 (VR1) and CB1 agonist/anandamide transport inhibitor
0462 (E)-Capsaicin
Prototypic vanilloid receptor agonist
1556 6'-Iodoresiniferatoxin
High affinity TRPV1 agonist/partial agonist
1568 NADA
Endogenous TRPV1 agonist. Also CB1 agonist
1641 OLDA
Potent, selective endogenous TRPV1 agonist
0934 Olvanil
Potent vanilloid receptor agonist
1466 PPAHV
Non-pungent vanilloid receptor agonist
1137 Resiniferatoxin
Potent vanilloid receptor agonist
3745 RN 1747
Selective TRPV4 agonist
Antagonists
Cat.No.
Product Name / Activity
4319 A 784168
Potent and selective TRPV1 antagonist
2316 AMG 9810
Potent and selective, competitive antagonist of TRPV1
2836 Arachidonyl serotonin
Dual FAAH inhibitor/TRPV1 antagonist
3875 BCTC
TRPV1 antagonist
0464 Capsazepine
Vanilloid receptor antagonist; also activator of ENaCδ
4100 HC 067047
Potent and selective TRPV4 antagonist
1975 6-Iodonordihydrocapsaicin
Potent, competitive vanilloid receptor antagonist
1362 5'-Iodoresiniferatoxin
Potent, silent TRPV1 antagonist
3361 JNJ 17203212
Reversible, competitive and potent TRPV1 antagonist
1577 L-R4W2
TRPV1 antagonist peptide
3746 RN 1734
Selective TRPV4 antagonist
1439 Ruthenium Red
Blocks capsaicin-activated cation channels
1615 SB 366791
Potent, selective, competitive TRPV1 antagonist
3265 SB 452533
Potent TRPV1 receptor antagonist
4729 α-Spinasterol
TRPV1 antagonist; active in vivo
1098 Tranilast
Antiallergic; inhibits TRPV2-mediated responses
Inhibitors
Cat.No.
Product Name / Activity
5106 GSK 2193874
Potent and selective TRPV4 inhibitor; orally active
Ligand Sets
Cat.No.
Product Name / Activity
2181 Vanilloid TRPV1 Receptor Tocriset™
Selection of 5 vanilloid TRPV1 receptor ligands (Cat. Nos. 0462, 0934, 1137, 0464 and 1615)
Other
Cat.No.
Product Name / Activity
4104 MM-22
Biotinylated anandamide analog; blocks anandamide uptake
2203 PALDA
Endogenous lipid; potentiates effects of endovanilloids at TRPV1 receptors
2204 STEARDA
Endogenous lipid, active in vivo. Enhances effects of endovanilloids at TRPV1 receptors
1684 Tocrisolve™ 100
Water-soluble emulsion; negative control for reagents in TocrisolveTM 100
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