5-HT₇ Receptors

More Information »Serotonin 5-HT₇ receptors are located primarily in the thalamus, hypothalamus and hippocampus. The function of these receptors includes the regulation of circadian rhythms, thermoregulation, learning and memory and smooth muscle relaxation.

5-HT₇ Receptor Products

Agonists
Cat.No.	Product Name / Activity
1968	AS 19
	Reported potent 5-HT₇ agonist
2925	LP 12 hydrochloride
	5-HT₇ agonist
2534	LP 44
	High affinity 5-HT₇ agonist
Antagonists
Cat.No.	Product Name / Activity
1523	LY 215840
	5-HT₂/5-HT₇ antagonist
2726	SB 258719 hydrochloride
	Selective 5-HT₇ antagonist
1612	SB 269970 hydrochloride
	Potent selective 5-HT₇ antagonist. Brain penetrant
Other
Cat.No.	Product Name / Activity
0458	5-Carboxamidotryptamine maleate
	Has high affinity for 5-ht_5A and 5-HT₇. Also 5-HT₁ agonist
0529	8-Hydroxy-DPAT hydrobromide
	Has moderate affinity for 5-HT₇. Also 5-HT_1A agonist
4704	LP 20 hydrochloride
	Selective 5-HT₇ ligand
0590	Metergoline
	Has moderate affinity for 5-HT₆ and high affinity for 5-HT₇. Also 5-HT₁/5-HT₂ antagonist
0937	Pimozide
	High affinity for 5-HT₇. Also D₂ antagonist

Related Categories

5-HT₁ Receptors 5-HT₂ Receptors 5-HT₄ Receptors

5-ht₅ Receptors 5-HT₆ Receptors

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5-HT Review

Written by Nicholas Barnes and John Neumaier, leading experts. Request a copy or view PDF today.

7-TM Receptor Signaling

Written by T. Kenakin et al

'Seven Transmembrane Receptor Signaling' highlights the multiple behaviors of 7-TMs including G-protein-dependent and -independent signaling as well as the concept of collateral efficacy