5-HT₄ Receptors

More Information »Serotonin 5-HT₄ receptors are located primarily in nigrostriatal and mesolimbic systems and smooth muscle. The receptor plays a role in memory and learning, anxiety, visual perception and smooth muscle relaxation.

5-HT₄ Receptor Products

Agonists
Cat.No.	Product Name / Activity
4374	BIMU 8
	Potent 5-HT₄ receptor full agonist
1695	Cisapride
	5-HT₄ agonist; stimulates intestinal ACh release
3089	CJ 033466
	Selective 5-HT₄ partial agonist
3499	ML 10302 hydrochloride
	Potent and selective 5-HT₄ partial agonist
2844	Mosapride citrate
	5-HT₄ agonist and 5-HT₃ antagonist
0736	2-[1-(4-Piperonyl)piperazinyl]benzothiazole
	5-HT₄ agonist. Also 5-HT₃ antagonist
0989	RS 67333 hydrochloride
	5-HT₄ partial agonist
0990	RS 67506 hydrochloride
	5-HT₄ partial agonist
4613	Tegaserod maleate
	5-HT₄ partial agonist
1795	Zacopride hydrochloride
	5-HT₄ agonist. Also highly potent 5-HT₃ antagonist
Antagonists
Cat.No.	Product Name / Activity
1322	GR 113808
	Potent, selective 5-HT₄ antagonist
1658	GR 125487 sulfamate
	Potent, selective 5-HT₄ antagonist. Active in vivo
0728	RS 23597-190 hydrochloride
	5-HT₄ antagonist
0991	RS 39604 hydrochloride
	5-HT₄ antagonist
0785	SB 203186 hydrochloride
	5-HT₄ antagonist
1373	SB 204070
	Potent and selective 5-HT₄ antagonist
2037	SDZ 205-557 hydrochloride
	5-HT₄/5-HT₃ receptor antagonist

Related Categories

5-HT₁ Receptors 5-HT₂ Receptors

5-ht₅ Receptors 5-HT₇ Receptors

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5-HT Review

Written by Nicholas Barnes and John Neumaier, leading experts. Request a copy or view PDF today.

7-TM Receptor Signaling

Written by T. Kenakin et al

'Seven Transmembrane Receptor Signaling' highlights the multiple behaviors of 7-TMs including G-protein-dependent and -independent signaling as well as the concept of collateral efficacy