R&D Systems Inc. Tocris Bioscience Boston Biochem

Melatonin Receptors

More Information »Melatonin receptors are a group of high affinity Gi/G0 protein-coupled receptors, which are split into two subtypes; MT1 and MT2. They are widely distributed with high concentrations found in the brain (especially in the suprachiasmatic nucleus) and in the retina.

Melatonin Receptor Products

Agonists
Cat.No.
Product Name / Activity
0357 N-Acetyltryptamine
Melatonin partial agonist (MT1/MT2). Also MT3 antagonist
0443 6-Chloromelatonin
Melatonin agonist
0737 2-Iodomelatonin
High affinity melatonin agonist
3550 Melatonin
Endogenous hormone; agonist at MT1 and MT2
1035 8-M-PDOT
Melatonin agonist
0680 2-Phenylmelatonin
Potent melatonin agonist
Antagonists
Cat.No.
Product Name / Activity
1218 DH 97
MT2 receptor antagonist
0877 Luzindole
Competitive melatonin MT1/MT2 antagonist
1034 4-P-PDOT
MT2 antagonist
0623 Prazosin hydrochloride
MT3 antagonist, also α1 and α2B antagonist
Ligands
Cat.No.
Product Name / Activity
0896 GR 135531
High affinity melatonin MT3 ligand

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7-TM Receptor Signaling

Written by T. Kenakin et al

7-TM Poster

'Seven Transmembrane Receptor Signaling' highlights the multiple behaviors of 7-TMs including G-protein-dependent and -independent signaling as well as the concept of collateral efficacy

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New Product Guide

NPG

Highlights 140 new products added in the first half of 2014. Request a copy or view PDF today.

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Human Proteome Organisation World Congress 2014

Human Proteome Organisation World Congress 2014

October 5 - 8, 2014

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