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Melatonin Receptors
More Information »Melatonin receptors are a group of high affinity Gi/G0 protein-coupled receptors, which are split into two subtypes; MT1 and MT2. They are widely distributed with high concentrations found in the brain (especially in the suprachiasmatic nucleus) and in the retina.
Melatonin Receptor Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 0357 | N-Acetyltryptamine |
| Melatonin partial agonist (MT1/MT2). Also MT3 antagonist | |
| 0443 | 6-Chloromelatonin |
| Melatonin agonist | |
| 0737 | 2-Iodomelatonin |
| High affinity melatonin agonist | |
| 3550 | Melatonin |
| Endogenous hormone; agonist at MT1 and MT2 | |
| 1035 | 8-M-PDOT |
| Melatonin agonist | |
| 0680 | 2-Phenylmelatonin |
| Potent melatonin agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 1218 | DH 97 |
| MT2 receptor antagonist | |
| 0877 | Luzindole |
| Competitive melatonin MT1/MT2 antagonist | |
| 1034 | 4-P-PDOT |
| MT2 antagonist | |
| 0623 | Prazosin hydrochloride |
| MT3 antagonist, also α1 and α2B antagonist | |
Ligands |
|
Cat.No. |
Product Name / Activity |
| 0896 | GR 135531 |
| High affinity melatonin MT3 ligand | |
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7-TM Receptor Signaling
Written by T. Kenakin et al
'Seven Transmembrane Receptor Signaling' highlights the multiple behaviors of 7-TMs including G-protein-dependent and -independent signaling as well as the concept of collateral efficacy
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