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Adrenergic β1 Receptors
More Information »The adrenergic β1 receptor (β1-adrenoceptor) is a member of the adrenergic receptor group of G-protein-coupled receptors that also includes α1A, α1B, α1D, α2A, α2B, α2C, β2 and β3. They are located primarily in the CNS, heart, coronary artery, kidney and muscle.
Adrenergic β1 Receptors Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 0950 | Xamoterol hemifumarate |
| β1 selective partial agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 0387 | (RS)-Atenolol |
| β1 antagonist | |
| 0393 | (S)-(-)-Atenolol |
| β1-antagonist. Active isomer of atenolol (Cat. No. 0387) | |
| 0906 | Betaxolol hydrochloride |
| Selective β1 antagonist | |
| 0914 | (±)-Bisoprolol hemifumarate |
| β1 antagonist | |
| 1024 | CGP 20712 dihydrochloride |
| Highly potent and selective β1 antagonist | |
| 3256 | Metoprolol tartrate |
| Selective β1 antagonist | |
| 3517 | Nebivolol hydrochloride |
| Highly selective β1-adrenoceptor antagonist | |
| 0649 | (S)-Timolol maleate |
| β1 antagonist | |
Ligand Sets |
|
Cat.No. |
Product Name / Activity |
| 1874 | β-Adrenoceptor Antagonist Tocriset™ |
| Selection of 3 β-adrenoceptor antagonists (Cat. Nos. 1024, 0821 and 1511) | |
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