Adenosine A1 Receptors

More Information »The A1 receptor is a member of the adenosine receptor group of G-protein-coupled receptors that also includes A2A, A2B and A3. A1 receptors display high expression levels in the brain (cortex, cerebellum, hippocampus), dorsal horn of the spinal cord, eye and atria.

A1 Receptor Products

Agonists
Cat.No.
Product Name / Activity
1705 2-Chloro-N6-cyclopentyladenosine
Potent, selective A1 agonist
1702 N6-Cyclopentyladenosine
Potent, selective A1 agonist
3576 (±)-5'-Chloro-5'-deoxy-ENBA
Highly selective A1 agonist
1957 GR 79236
A1 agonist
2281 2'-MeCCPA
Very selective and potent A1 receptor agonist
2465 SDZ WAG 994
Potent, selective A1 agonist
Antagonists
Cat.No.
Product Name / Activity
0486 1,3-Dipropyl-8-phenylxanthine
A1 selective antagonist
0439 DPCPX
A1 selective antagonist
4167 KW 3902
Selective A1 antagonist
2019 PSB 36
Potent and selective A1 antagonist
3344 SLV 320
Potent and selective A1 antagonist
Modulators
Cat.No.
Product Name / Activity
1363 PD 81723
Allosteric potentiator of A1 receptors
Controls
Cat.No.
Product Name / Activity
5122 Dansyl-NECA
Potent and selective fluorescent adenosine A1 agonist
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