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Adenosine A1 Receptors
More Information »The A1 receptor is a member of the adenosine receptor group of G-protein-coupled receptors that also includes A2A, A2B and A3. A1 receptors display high expression levels in the brain (cortex, cerebellum, hippocampus), dorsal horn of the spinal cord, eye and atria.
A1 Receptor Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 1705 | 2-Chloro-N6-cyclopentyladenosine |
| Potent, selective A1 agonist | |
| 1702 | N6-Cyclopentyladenosine |
| Potent, selective A1 agonist | |
| 3576 | (±)-5'-Chloro-5'-deoxy-ENBA |
| Highly selective A1 agonist | |
| 1957 | GR 79236 |
| A1 agonist | |
| 2281 | 2'-MeCCPA |
| Very selective and potent A1 receptor agonist | |
| 2465 | SDZ WAG 994 |
| Potent, selective A1 agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 0486 | 1,3-Dipropyl-8-phenylxanthine |
| A1 selective antagonist | |
| 0439 | DPCPX |
| A1 selective antagonist | |
| 4167 | KW 3902 |
| Selective A1 antagonist | |
| 2019 | PSB 36 |
| Potent and selective A1 antagonist | |
| 3344 | SLV 320 |
| Potent and selective A1 antagonist | |
Modulators |
|
Cat.No. |
Product Name / Activity |
| 1363 | PD 81723 |
| Allosteric potentiator of A1 receptors | |
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7-TM Receptor Signaling
Written by T. Kenakin et al
'Seven Transmembrane Receptor Signaling' highlights the multiple behaviors of 7-TMs including G-protein-dependent and -independent signaling as well as the concept of collateral efficacy
Regulation of Vascular Reactivity by GPCRs
Written by J.J. Maguire and A.P. Davenport
'Regulation of Vascular Reactivity by G-protein-coupled Receptors' summarizes the key GPCRs regulating vascular reactivity.
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