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M1 Receptors
More Information »M1 receptors are members of the G-protein-coupled receptor (GPCR) family which are found mostly bound to Gq proteins. They are one of five muscarinic receptors that act to control the metabotropic functions of acetylcholine (ACh) in the central nervous system (CNS).
M1 Receptor Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 3689 | Cevimeline hydrochloride |
| Selective M1 agonist | |
| 1384 | McN-A 343 |
| Selective M1 muscarinic agonist | |
| 3569 | Xanomeline oxalate |
| Functionally selective M1 agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 2853 | Biperiden hydrochloride |
| Muscarinic receptor antagonist; some selectivity for M1 | |
| 0469 | Nitrocaramiphen hydrochloride |
| Muscarinic antagonist, M1 > M2 | |
| 1071 | Pirenzepine dihydrochloride |
| Selective M1 muscarinic antagonist | |
| 1122 | Telenzepine dihydrochloride |
| Potent, selective M1 antagonist | |
| 3727 | VU 0255035 |
| Highly selective muscarinic M1 antagonist | |
Modulators |
|
Cat.No. |
Product Name / Activity |
| 4295 | VU 0357017 hydrochloride |
| Positive allosteric modulator of M1 receptors | |
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