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Aryl Hydrocarbon Receptors

More Information »Aryl hydrocarbon receptors (AHRs) are cytosolic transcription factors that exist bound to co-chaperones in the resting state. Ligand binding causes the co-chaperones to dissociate, allowing AHR to translocate to the nucleus, dimerize and alter transcription of target genes.

Aryl Hydrocarbon Receptor Products

Agonists
Cat.No.	Product Name / Activity
1803	ITE
	Endogenous agonist for the transcription factor aryl hydrocarbon receptor
3873	MeBIO
	AhR agonist. Inactive analog of BIO (Cat. No. 3194)
1267	Pifithrin-α hydrobromide
	Aryl hydrocarbon receptor agonist. Also p53 inhibitor
Antagonists
Cat.No.	Product Name / Activity
3858	CH 223191
	Potent aryl hydrocarbon receptor (AhR) antagonist
3859	6,2',4'-Trimethoxyflavone
	Aryl hydrocarbon receptor antagonist
Modulators
Cat.No.	Product Name / Activity
4628	DiMNF
	Selective aryl hydrocarbon receptor modulator (SAhRM)
Ligands
Cat.No.	Product Name / Activity
4393	L-Kynurenine
	Tryptophan catabolite; endogenous aryl hydrocarbon receptor ligand

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