Histone Methyltransferases

More Information »Histone methyltransferases (HMTs) are a group of enyzmes that catalyze the transfer of methyl groups from S-adenosylmethionine (SAM) to histones. This occurs predominantly on the side chains of lysine and arginine residues in histones H3 and H4.

Histone Methyltransferase Products

Inhibitors
Cat.No.
Product Name / Activity
5163 A 366
Potent and selective G9a/GLP inhibitor
3364 BIX 01294
GLP and G9a inhibitor
5128 C 21
Selective PRMT1 inhibitor
4504 Chaetocin
SUV39H1 inhibitor
4703 3-Deazaneplanocin A hydrochloride
Histone methyltransferase inhibitor
5567 EPZ 004777
Highly potent DOT1L inhibitor
5202 Furamidine dihydrochloride
Selective PRMT1 inhibitor
4892 (R)-PFI 2 hydrochloride
Potent and selective SETD7 inhibitor
5400 (S)-PFI 2 hydrochloride
Negative control of (R)-PFI 2 hydrochloride (Cat. No. 4892)
2609 Ryuvidine
SETD8 inhibitor; also CDK4 inhibitor
4541 SGC 0946
Highly potent and selective DOT1L inhibitor; cell permeable
5367 SGC 707
Potent and selective allosteric inhibitor of PRMT3
5099 TC-E 5003
Selective PRMT1 inhibitor
3861 UNC 0224
Potent G9a inhibitor
4343 UNC 0638
Selective G9a and GLP inhibitor
5132 UNC 0642
Potent and selective G9a and GLP inhibitor
4342 UNC 0646
Potent and selective G9a/GLP inhibitor
4904 UNC 1999
Potent and selective EZH2/EZH1 inhibitor
5057 UNC 2327
Allosteric inhibitor of PRMT3
4905 UNC 2400
Negative control of UNC 1999 (Cat. No. 4904)
5450 XY1
Negative control of SGC 707 (Cat. No. 5367)
Other
Cat.No.
Product Name / Activity
5307 MM 102
WDR5/MLL interaction inhibitor
5267 OICR 9429
High affinity and selective WDR5 antagonist
5323 WDR5 0103
WDR5 antagonist
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