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5-HT2C Receptors
More Information »Serotonin 5-HT2C receptors, previously known as 5-HT1C receptors, are located primarily in the choroid plexus, cortex, limbic system and basal ganglia. 5-HT2C receptors play a role in CSF volume regulation, thermoregulation, penile erection and anxiety.
5-HT2C Receptor Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 3041 | CP 809101 hydrochloride |
| Potent and selective 5-HT2C agonist | |
| 0875 | m-CPP hydrochloride |
| 5-HT2B/2C receptor agonist | |
| 2643 | DOI hydrochloride |
| Mixed 5-HT2A/2C agonist | |
| 1860 | Eltoprazine hydrochloride |
| 5-HT2C receptor partial agonist | |
| 3017 | 1-Methylpsilocin |
| Potent and selective 5-HT2C agonist | |
| 0941 | MK 212 hydrochloride |
| 5-HT2C agonist | |
| 3585 | Org 12962 hydrochloride |
| Selective 5-HT2C agonist | |
| 2201 | PNU 22394 hydrochloride |
| 5-HT2C agonist and 5-HT2A/2B partial agonist | |
| 1854 | Ro 60-0175 fumarate |
| Potent, selective 5-HT2C agonist | |
| 0925 | SCH 23390 hydrochloride |
| 5-HT2C agonist. Also potent dopamine D1-like antagonist | |
| 1801 | WAY 161503 hydrochloride |
| Potent, selective 5-HT2C agonist | |
| 2173 | WAY 629 hydrochloride |
| Selective 5-HT2C agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 0444 | Clozapine |
| 5-HT2A/2C antagonist. Also dopamine antagonist | |
| 1007 | N-Desmethylclozapine |
| 5-HT2C antagonist | |
| 1644 | Mesulergine hydrochloride |
| 5-HT2A and 5-HT2C antagonist. Also dopamine receptor partial agonist | |
| 1050 | RS 102221 hydrochloride |
| Selective 5-HT2C antagonist | |
| 4508 |
S 32212 hydrochloride
|
| 5-HT2C inverse agonist; α2 antagonist | |
| 1371 | SB 200646 hydrochloride |
| 5-HT2C/2B antagonist | |
| 1661 | SB 206553 hydrochloride |
| Potent, selective 5-HT2C/5-HT2B antagonist. Orally active | |
| 1379 | SB 221284 |
| Potent, selective 5-HT2C/2B antagonist | |
| 1375 | SB 228357 |
| 5-HT2C/2B antagonist/inverse agonist | |
| 2901 | SB 242084 |
| Selective 5-HT2C antagonist; brain penetrant | |
| 3527 | SB 243213 dihydrochloride |
| Selective 5-HT2C inverse agonist | |
| 1255 | SDZ SER 082 fumarate |
| Selective 5-HT2B/2C antagonist | |
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