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Purinergic (P2Y) Receptors
More Information »P2Y receptors are G-protein-coupled receptors that respond to extracellular purine and pyrimidine nucleotides. To date, eight mammalian P2Y receptors are known (P2Y1, P2Y2, P2Y4, P2Y6, P2Y11-14) as well as the non-mammalian p2y3, p2y8 and p2y receptors.
Purinergic (P2Y) Receptor Products
Agonists |
|
Cat.No. |
Product Name / Activity |
| 3245 | ATP disodium salt |
| P2 agonist | |
| 4080 | ATPγS tetralithium salt |
| P2 agonist; ATP (Cat. No. 3245) analog | |
| 3312 | BzATP triethylammonium salt |
| P2Y1 partial agonist. Also P2X7 agonist and P2X1 partial agonist | |
| 3209 | α,β-Methyleneadenosine 5'-triphosphate trisodium salt |
| P2 agonist | |
| 1624 | 2-Methylthioadenosine diphosphate trisodium salt |
| Potent agonist for P2Y1, P2Y12 and P2Y13 | |
| 1062 | 2-Methylthioadenosine triphosphate tetrasodium salt |
| P2 agonist | |
| 2157 | MRS 2365 |
| Highly potent and selective P2Y1 agonist | |
| 2915 | MRS 2690 |
| Potent P2Y14 agonist | |
| 2502 | MRS 2693 trisodium salt |
| Selective P2Y6 agonist | |
| 3884 | MRS 2768 tetrasodium salt |
| Selective P2Y2 agonist | |
| 4260 | MRS 2957 triethylammonium salt |
| Potent and selective P2Y6 agonist | |
| 4261 | MRS 4062 triethylammonium salt |
| Selective P2Y4 receptor agonist | |
| 3892 | NF 546 |
| Selective P2Y11 agonist | |
| 4376 | 5-OMe-UDP trisodium salt |
| Potent P2Y6 agonist | |
| 2715 | PSB 0474 |
| Potent and selective P2Y6 agonist | |
| 4333 | PSB 1114 |
| Potent, selective P2Y2 agonist | |
| 3280 | 2-ThioUTP tetrasodium salt |
| Potent and selective P2Y2 agonist | |
| 3279 | UTPγS trisodium salt |
| Selective P2Y2/4 agonist | |
Antagonists |
|
Cat.No. |
Product Name / Activity |
| 3321 | AR-C 66096 tetrasodium salt |
| Potent and selective P2Y12 antagonist | |
| 1820 | (+)-Clopidogrel hydrogen sulfate |
| Selective P2Y12 antagonist | |
| 2490 | (±)-Clopidogrel hydrochloride |
| Selective P2Y12 antagonist | |
| 0900 | MRS 2179 tetrasodium salt |
| Selective P2Y1 antagonist | |
| 2402 | MRS 2211 |
| Competitive P2Y13 antagonist | |
| 2158 | MRS 2279 |
| Selective, high affinity P2Y1 antagonist | |
| 2159 | MRS 2500 tetraammonium salt |
| Extremely potent and selective P2Y1 antagonist | |
| 2146 | MRS 2578 |
| Selective P2Y6 antagonist | |
| 2450 | NF 157 |
| Selective P2Y11/P2X1 antagonist | |
| 3830 | NF 340 |
| Selective P2Y11 antagonist | |
| 0625 | PPADS tetrasodium salt |
| P2 antagonist | |
| 3983 | PSB 0739 |
| Highly potent P2Y12 receptor antagonist | |
| 1472 | Suramin hexasodium salt |
| Non-selective P2 antagonist | |
| 3931 | Ticlopidine hydrochloride |
| Selective P2Y12 antagonist | |
Other |
|
Cat.No. |
Product Name / Activity |
| 1682 | PIT |
| P2Y ligand; displays mixed antagonism/potentiation | |
| 3111 | UDP disodium salt |
| Endogenous ligand; competitive antagonist at P2Y14 receptors | |
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