All Products

Cat.No.

Product Name / Activity

Selective p300/CBP HAT inhibitor

Adenine receptor agonist

MIF binder

CB₂ agonist

Selective and potent COX-2 inhibitor

Selective D₃ antagonist

High affinity 5-HT₆ antagonist

Selective 5-HT₆ agonist

Calcineurin phosphatase inhibitor; analog of FK 506 (Cat. No. 3631)

Negative control of IPA 3 (Cat. No. 3622)

Potent and selective CCR3 antagonist

Naturally-occurring prostanoid; potent vasoconstrictor

Protein translation inhibitor; blocks eIF4F subunit interaction

High affinity, selective AT₁ antagonist

Potent and selective FP prostaglandin receptor agonist

Prodrug topoisomerase II inhibitor

Adenosine receptor antagonist

Potent JAK3 inhibitor. Also inhibits GSK-3β and PKC

Dynamin I inhibitor

Dynamin inhibitor

Dynamin inhibitor

Inhibitor of LFA-1/ICAM mediated cell adhesion

Potent inhibitor of the LFA-1/ICAM-1 interaction

Caged D-AP5 (Cat.No. 0106)

K_ir6 (K_ATP) blocker; displays high affinity for SUR1/K_ir6.2 channels

Potent P2X₇ antagonist

Positive allosteric modulator of α7 nAChRs

CB₁ receptor antagonist

Selective MEK inhibitor

Potent and selective IKKβ inhibitor

Highly selective c-Met inhibitor

H₁ antagonist; ocular antiallergic agent

MCH₁ antagonist

Endogenous ligand for KISS1 receptor

Human pregnane X receptor agonist; H₁ antagonist

Selectively inhibits PKC-induced NF-κB activation

Potent and selective mTOR inhibitor

Potent and selective mTOR inhibitor

Potent voltage-dependent Na_V1.8 channel blocker

Topoisomerase II inhibitor; immunosuppressive and antineoplastic agent

Selective CYP3A4 inhibitor

Inhibitor of human telomerase

Potent p38 MAPK inhibitor; anti-inflammatory

Potent and selective GPR139 agonist

GABA uptake inhibitor; anticonvulsant

Dual mTORC1/mTORC2 inhibitor

Positive allosteric modulator of mGlu₄

Potent and selective P2Y₆ agonist

Selective P2Y₄ receptor agonist

Selective, potent inhibitor of CLK1 and 4

PI 3-kinase inhibitor

Selective inhibitor of Cdc42 Rho family GTPase

Class I histone deacetylase inhibitor

Selective MC₃ receptor agonist

Potent and selective LRRK2 inhibitor

Potent multi-kinase and pan-BCR-ABL inhibitor

Potent ERβ agonist

Selective Chk1 inhibitor

Dual FAK/PYK2 inhibitor

Potent MK2 inhibitor

Selective casein kinase 1ε inhibitor

Potent and selective mTOR inhibitor

γ-secretase inhibitor; lowers Aβ40 and Aβ42 levels

Selective USP7 inhibitor

Inhibits microtubule polymerization

TLR3 agonist

Potent S1P₁ agonist

Potent pan-Aurora kinase inhibitor

Potent and selective PLK1 inhibitor

GPR35 antagonist

Selective farnesyltransferase (FTase) inhibitor

Positive allosteric modulator of M₁ receptors

Positive regulator of autophagy

GPR35 agonist

Inhibits β-catenin-responsive transcription (CRT)