All Products

Cat.No.

Product Name / Activity

α₄β₁ (VLA-4) antagonist

Control peptide for neuropeptide Y (Cat. No. 1173)

Selective 5-HT₆ agonist

Ca²⁺ mobilizing agent

Antitumor and anti-HIV agent; activates NF-κB. Also TGR5 agonist

Selective α₄β₁ (VLA-4) inhibitor

Positive allosteric modulator of AMPA

RXR antagonist

RXR synergist

Inhibitor of Src family kinases

Potent and selective p38α inhibitor

Orally active p38α and p38β inhibitor

Antibiotic; inhibits protein, DNA and RNA synthesis in gram-positive bacteria

Potent inhibitor of multi-drug and toxin extrusion (MATE) transporters; also inhibits DHFR

Selective cyclooxygenase-2 (COX-2) inhibitor

Potent and selective p38α inhibitor

High affinity CB₁ antagonist

Potent inhibitor of ER-associated protein degradation and translocation

Non-steroidal androgen receptor antagonist

Orally active vasopressin V₁ antagonist

Selective ERRα antagonist/inverse agonist

MDMX inhibitor. Disrupts MDMX-p53 interaction

Inhibitor of calcineurin-mediated NFAT activation

Selective P2Y₁₂ antagonist

Potent NOP agonist; displays analgesic properties

Potent non-peptide oxytocin receptor agonist

Calcium channel blocker

α_2D agonist

Potent and selective PDE4 inhibitor

Adenosine A_2A antagonist

TRPA1 blocker

Inhibitor of SOCE in non-excitable cells

D₃ antagonist. Also D₂ partial agonist

Subtype-selective GABA_A receptor agonist

GABA_A α2 benzodiazepine receptor agonist

CFTR mutants potentiator

Neuroprotective peptide; protects against β-amyloid neurotoxicity

Inhibitor of IP6K; also inhibits IP3K

Negative control for endo-IWR 1 (Cat. No. 3532)

H₁ antagonist. Also K_V11.1 (hERG) and K_ir6 (K_ATP) channel blocker

Positive allosteric modulator of mGlu₂

Arp2/3 inhibitor; inhibits actin polymerization

Potent CXCR4 antagonist

NAADP antagonist; inhibits Ca²⁺ release

NAADP antagonist; inhibits Ca²⁺ release

μ-opioid receptor agonist

Ghrelin receptor (GHS-R1a) antagonist

Potent, selective and reversible CerK inhibitor

Potent and selective PPARδ antagonist

Selective PKD inhibitor; analog of CID 755673 (Cat. No. 3327)

Src tyrosine kinase inhibitor

α7-selective agonist

PPARα/γ agonist

Selective GSK-3 inhibitor

Allosteric glycogen phosphorylase inhibitor

Potent cyclin-dependent kinase (cdk) 1, 2 and 9 inhibitor

Selective iNOS inhibitor

Active metabolite of vitamin D₂

Deuterated nalmefene; opioid receptor antagonist

Positive allosteric modulator of GABA_A receptors

Inhibitor of actin assembly and polymerization

Estrogen receptor ligand; mycotoxin

Mycotoxin; potent protein synthesis inhibitor

Class III PI 3-kinase inhibitor; also inhibits autophagy

Selective B₂ antagonist; analog of HOE 140 (Cat. No. 3014)

Selective inhibitor of PTPMT1

Dynamin inhibitor; attenuates mitochondrial division and apoptosis

Highly potent P2Y₁₂ receptor antagonist

MDM2 antagonist; inhibits MDM2-p53 interaction

β3 agonist; displays anxiolytic and antidepressant effects

Potent Aurora kinase B inhibitor

TRPM8 blocker

Caged noradrenalin

Caged serotonin

Caged dopamine

Vitamin D receptor (VDR) agonist

Potent and selective monopolar spindle 1 (Mps1) kinase inhibitor

5-HT_2A/D₂ antagonist; atypical antipsychotic

Receptor-selective retinoid; binds RAR-β and -γ

Ubiquitin C-terminal hydrolase-L1 (UCH-L1) inhibitor

Selective estrogen receptor modulator (SERM)