All Products

Cat.No.

Product Name / Activity

Potent FGFR and VEGFR inhibitor

Cyclin-dependent kinase 2 (cdk2) inhibitor

Potent and selective RXRα agonist.

RXR antagonist

Potent and selective PDGFRβ inhibitor

Uroselective α₁ antagonist

Selective A_2A antagonist. Also MAO-B inhibitor

Selective FAAH inhibitor

Orally active 5-LOX inhibitor

HMG-CoA reductase inhibitor

Potent, positive allosteric mGlu₄ agonist. Sodium salt of VU 0155041 (Cat. No. 3248)

P2X₇ agonist. Also P2X₁ and P2Y₁ partial agonist

Potent, selective GABA_B positive allosteric modulator

Selective, competitive JNK inhibitor

Potent PDE4 inhibitor

Potent and selective CK1ε and CK1δ inhibitor

Potent and selective human P2X₇ antagonist

IKKβ inhibitor; attenuates NF-κB-induced gene expression

Selective nNOS inhibitor

Potent and selective P2Y₁₂ antagonist

Potent P2X₇ receptor antagonist

ARFGAP1 inhibitor; modulates Wnt/β-catenin signaling

mGlu₅ positive allosteric modulator

High affinity 5-HT₆ antagonist

Selective protein kinase D inhibitor

Positive allosteric modulator of α4β2

Potent, competitive MAGL inhibitor

Caged (S)-3,4-DCPG

Caged (1S,3R)-ACPD

Caged group II mGlu receptor agonist

Potent, selective human C5a receptor antagonist

PDGFR, VEGFR and FGFR inhibitor

Potent AMPK activator

Neuromodulating neuropeptide fragment; satiety factor

Neuromodulatory neuropeptide fragment; satiety factor

Neuromodulating neuropeptide fragment; inhibits food intake in vivo

Alcohol dehydrogenase 7 inhibitor; inhibits downstream Hh signaling pathway

Potent and highly selective EP₃ antagonist

Selective NR2B antagonist

Potent and selective A₁ antagonist

MCH₁ antagonist; also 5-HT_2B antagonist and partial antagonist of 5-HT_1A

Potent and selective MCH₁ antagonist

Panx-1 mimetic inhibitory peptide; blocks pannexin-1 gap junctions

Versatile marker for neuroanatomical investigations

Dual 5-HT_1B/1D antagonist and 5-HT re-uptake inhibitor

Potent ErbB receptor family inhibitor

GPR119 receptor agonist

Competitive inhibitor of SREBP site 1 protease

Highly selective D₃ antagonist

p53 activator. Also ROS scavenger

Antitumor and intercalating agent; inhibits DNA topoisomerase II

Calpain inhibitor; activates p53-dependent apoptosis

Potent and selective MCH₁ antagonist

EGFR inhibitor. Also inhibits Aβ42 fibril formation

Reversible, competitive and potent TRPV1 antagonist

Restores mutant p53 activity; proapoptotic

G9a-like protein and G9a histone lysine methyltransferase inhibitor

Protects against MDM2-mediated p53 degradation

Selective ERβ agonist

Downregulates Bcl-2 and Mcl-1; pro-apoptotic

Orally active, selective 5-HT₆ antagonist

Potent and selective PAR₂ agonist

PAR₂ receptor agonist

Potent and selective OX₂ antagonist

Selective K⁺ ionophore

Endogenous neuropeptide; binds sst₁ - sst₅ and GHS-R1a

Selective vasopressin V_1A antagonist

Inhibits TRPP3-mediated currents; also inhibits the Na⁺/H⁺ exchanger (NHE)

Inhibits TRPP3-mediated currents; also inhibits epithelial Na⁺ channels

NCX inhibitor, Deg/ENaC channel blocker; amiloride (Cat. No. 0890) derivative

Anandamide uptake inhibitor. Also FAAH inhibitor and CB receptor partial agonist

Positive allosteric modulator of M₄ receptors

O-GlcNAcase and β-hexosaminidase inhibitor

P2X₇ allosteric modulator

Hsp90 inhibitor; exhibits anticancer and antimalarial activity

Potent aromatase (CYP19) inhibitor

Non-steroidal androgen receptor antagonist

Potent actin polymerization regulator

Inactive control peptide for amyloid β-peptide (1-42) (Cat. No. 1428)

Control peptide for SLIGKV-NH₂ (Cat. No. 3010)

Control peptide for TFLLR-NH₂ (Cat. No. 1464)

Control peptide for SLIGRL-NH₂ (Cat. No. 1468)

JAK2, FLT3 and TrkA inhibitor

Synthetic vasopressin analog; V_1B and V₂ agonist

Potent and selective GlyT1 inhibitor

Major antigenic component implicated in the pathophysiology of multiple sclerosis