All Products

Cat.No.

Product Name / Activity

CB₁/CB₂ receptor partial agonist

Non-competitive mGlu₁ antagonist with inverse agonist activity

Selective P2Y₆ agonist

Water-soluble GABA_A antagonist

PDE4 inhibitor; antiulcer agent

Monovalent cation ionophore

Potent, orally active human leukocyte elastase inhibitor

Potent, selective M₃ antagonist

Potent and selective NOP antagonist

Inhibitor of NF-κB activation; anti-inflammatory

CaCC blocker and Cl^-/HCO₃^- exchange)

Tryptase inhibitor

Endothelin-converting enzyme (ECE) inhibitor

Inhibits viral DNA polymerase; antiherpetic agent

Selective EP₄ receptor antagonist

Highly selective CCR2 chemokine receptor antagonist

α7-selective agonist

GnRH receptor antagonist

Broad spectrum MMP inhibitor

Histone deacetylase inhibitor

Secretory phospholipase A₂ (sPLA₂) inhibitor

Selective inhibitor of E-selectin and ICAM-1 expression

Urotensin-II (UT) antagonist

Subtype-selective NR2C/NR2D antagonist

Potent, positive allosteric modulator of GABA_A receptors

High affinity EAAT1 and EAAT2 blocker

Blocker of K_V1.5 channel and I_Kur current

High affinity 5-HT₇ agonist

Peripheral D₂-like antagonist

Neurotoxic amino acid

Selective inhibitor of IKK

Novel fluorescent cannabinoid ligand. Fluorescent form of AM 251 (Cat. No. 1117)

Potent, selective VEGFR-2 inhibitor

GnRH receptor agonist

5-HT and noradrenalin re-uptake inhibitor (SNRI)

Cell-permeable protein kinase A inhibitor

Selective catecholaminergic neurotoxin

Potent P2X₃ antagonist

Cell-permeable inhibitor of atypical PKC isozyme PKMζ

Non-peptide calcitonin (CT) receptor agonist

Vitamin D receptor (VDR) agonist

Potent and selective RARγ agonist

Non-competitive AMPA receptor antagonist

Potent and selective 5-HT_1D agonist

Non-competitive NMDA receptor antagonist

Selective Akt/PKB inhibitor

Potent, selective inhibitor of IKKβ

Inhibitor of checkpoint kinase 1 (Chk1)

Calmodulin antagonist

High affinity σ₂ agonist

Potent, selective farnesoid X receptor (FXR) agonist

20S proteasome inhibitor

Selective, non-peptide CCR8 agonist

High affinity melanocortin receptor agonist

Encephalitogenic myelin proteolipid fragment

Encephalitogenic myelin oligodendrocyte glycoprotein fragment

Selective, high affinity AT₂ ligand

Endogenous ligand for KISS1 receptor (hOT7T175/AXOR12/GPR54)

Ca²⁺ channel blocker (L-type)

Non-selective NTPDase inhibitor

NTPDase 3 inhibitor

Inhibits multiple neurotensin and neuromedin N degrading enzymes

Endogenous, selective NK₁ agonist

Selective H₁ antagonist

Angiotensin-converting enzyme (ACE) inhibitor

Selective M₃ antagonist

NSAID, cyclooxygenase (COX-1) inhibitor. Also opener of K_IR2.3

Activator of procaspase-3; pro-apoptotic

H⁺,K⁺-ATPase inhibitor

H⁺,K⁺-ATPase inhibitor

Endogenous melanocortin receptor agonist

C3-binding protein, inhibits complement activation

Soluble guanylyl cyclase (sGC) activator

Potent FLT3 inhibitor

Potent, high affinity 5-HT_2A agonist

Potent CCR1 chemokine receptor antagonist

Na⁺ channel blocker, antiarrhythmic agent

Potent and selective NOP antagonist

Dopamine stabilizer