All Products

Cat.No.

Product Name / Activity

High affinity NK₁ receptor antagonist

Competitive P2Y₁₃ antagonist

High affinity, selective A₃ antagonist

Na⁺ channel blocker

Farnesyltransferase (FTase) inhibitor; antitumor

Prodrug form of FTI 276 (Cat. No. 2406)

Inhibitor of Aβ42 fibril formation

Potent and selective H₃ receptor antagonist

Potent and selective oxytocin receptor antagonist

Potent and selective CCK₁ agonist. Suppresses feeding

Highly selective NPY Y₁ receptor antagonist

Selective Rho-kinase (ROCK) inhibitor

Cell-permeable, selective Rho-kinase inhibitor

Highly selective EGFR-kinase inhibitor

Selective inhibitor of EGFR-kinase

Negative control of LY 294002 (Cat. No. 1130)

Selective H₃ antagonist

Potent peptide agonist for APJ receptor

Histone deacetylase inhibitor

Akt/PKB substrate (synthetic)

Chemokine receptor 5 (CCR5) antagonist

Amyloid β-protein fragment

Predominant amyloid β-protein fragment

Endogenous APJ receptor agonist

Endogenous APJ receptor agonist

H₁ receptor antagonist; non-sedating antiallergic agent

Geranylgeranyltransferase I (GGTase I) inhibitor

Potent PDE3 inhibitor

High affinity, selective CB₂ agonist

Highly selective CB₂ agonist

Hsp90 inhibitor

Selective RARβ2 agonist

Neuronal nicotinic receptor antagonist

Selective sst₄ agonist

Selective H₄ receptor antagonist; orally active

Selective inhibitor of PKCβII

MDM2-p53 interaction inhibitor

Potent and selective sst₂ agonist

Endogenous anorexigenic peptide

Immunomodulator; inhibits IL-10 synthesis and potentiates IL-1α, IL-2 and TNF-α release

Derivative of mGlu₁ antagonist YM 298198 (Cat. No. 2448)

Highly potent, selective non-competitive mGlu₁ antagonist

Selective P2Y₁₁/P2X₁ antagonist

Potent, selective 5-HT_1F agonist

Novel, potent anandamide uptake inhibitor. Inhibits FAAH

Highly selective group II mGlu agonist

Potent and selective sst₁ receptor agonist

Highly selective NR2B antagonist

Potent cdk4/cyclin D1 and CaM Kinase II inhibitor. Antiviral agent (anti-HCMV)

Inhibits Aurora kinase B

Potent 5-HT₃ receptor antagonist; orally active

Selective MAO-B inhibitor

Very selective, high affinity A_2A antagonist

Potent, selective P2X antagonist

Potent, selective A₁ agonist

α₂ agonist. Water-soluble form of UK 14,304 (Cat. No. 0425)

Selective central benzodiazepine receptor partial agonist

Selective agonist for the GPR109B (HM74) receptor. Antilipolytic

Cyclooxygenase-2 (COX-2) inhibitor

Selective Syk kinase inhibitor

Selective farnesoid X receptor (FXR) agonist

Orally active liver X receptor (LXR) agonist

Potent, selective inhibitor of VEGFR-2

Inhibitor of AP-1 transcription factor; antitumor agent

High affinity H₃ ligand

H₁ receptor agonist

Selective CB₂ receptor antagonist/inverse agonist

Selective NOP antagonist

Inhibitor of human telomerase activity

Non-peptide UT receptor agonist

Selective Rho-kinase (ROCK) inhibitor. More selective analog of H 1152 dihydrochloride (Cat. No. 2414)

Potent fatty acid synthase inhibitor; proapoptotic

Selective P2Y₁₂ antagonist

Orally active, high affinity 5-HT_1A agonist

Novel, non-toxic immunosuppressive agent

Potent H₃ receptor silent antagonist

Potent, high affinity H₄ agonist

5-HT_2A/D₂ receptor antagonist; neuroleptic

PARP-1 and PARP-2 inhibitor

Positive allosteric modulator of α7 nAChR; active in vivo

Inhibitor of VEGF receptor tyrosine kinase