All Products

Cat.No.

Product Name / Activity

Non-selective NOS inhibitor. Sodium salt of 7-nitroindazole (Cat. No. 0602)

Specific group III mGlu antagonist

Selective group I mGlu agonist. Active enantiomer of 3,5-DHPG (Cat. No. 0342)

Anticonvulsant. Increases brain GABA

GABA_A agonist

GABA-T inhibitor

EAAT2 and EAAT4 blocker

Weak NMDA antagonist

δ selective peptide antagonist

Very selective β₂ antagonist

κ agonist, acts peripherally

PPAR agonist

PPAR agonist

Potent, selective H₂ antagonist

δ selective peptide antagonist

β antagonist

Potentiates GABA_A receptor function

β antagonist

Potent H₂ antagonist, active in vivo

β antagonist. More active enantiomer of propranolol (Cat. No. 0624)

β antagonist. Less active enantiomer of propranolol (Cat. No. 0624)

Potent thromboxane receptor antagonist

Potent thromboxane A₂/TP receptor antagonist

Ca²⁺ release inhibitor

Peripherally acting μ agonist. Also Ca²⁺ channel blocker

High affinity ligand (σ₁ = σ₂)

α₂ ligand. Also imidazoline ligand

Muscarinic agonist

Potent inhibitor of L-glutamate uptake into synaptic vesicles

Potent inhibitor of L-glutamate uptake into synaptic vesicles; also inhibits MIF

Propranolol (Cat. No. 0624) metabolite

Group III/group II mGlu antagonist. More selective for group III than group II

Group II/group III mGlu antagonist

Group II/group III mGlu antagonist. More selective for group II than group III

5-HT_1D agonist

Desensitization inhibitor (AMPA > kainate)

Potent, selective NK₁ antagonist

NMDA antagonist, acts glycine site

5-HT_2A antagonist

Potent, selective iNOS inhibitor

Selective iNOS inhibitor, acts arginine binding site

5-HT_2B/2C receptor agonist

K_V channel blocker

Competitive melatonin MT₁/MT₂ antagonist

CB₁ receptor agonist

Selective GPR55 agonist. FAAH and PAA substrate

Selective inhibitor of NO-sensitive guanylyl cyclase

Potentiates GABA_A receptor function

Kir6 (K_ATP) channel opener

Selective σ₁ ligand, putative antagonist

Selective D₁-like agonist

α₂ agonist. Also I₂ selective ligand

Selective α₁ agonist

High affinity I₂ ligand. Highly selective

Na⁺ channel blocker. Also I₂ imidazoline ligand

α₂ antagonist

Standard δ₂ selective antagonist

Standard selective D₂-like antagonist

Standard selective D₂-like antagonist

High affinity melatonin MT₃ ligand

iNOS inhibitor, acts at arginine binding site

Irreversible μ antagonist

Standard δ₁ selective antagonist