All Products

Cat.No.

Product Name / Activity

Highly potent 5-HT₃ receptor antagonist. Also 5-HT₄ agonist

Benzodiazepine site agonist

Selective M₃ antagonist

Agonist at 'low affinity' GABA_A receptor. More potent than GABA/muscimol

PDE5/6/9/11 inhibitor

PDE3/4 inhibitor

Bradycardic agent; blocks I_f pacemaker current

Group III mGlu agonist (mGlu₄ > mGlu₈ > mGlu₇)

β₃-adrenoceptor agonist

β₃ agonist

Selective non-peptide AT₁ antagonist

Sino-atrial node function modulator (I_f inhibitor)

DNA methyltransferase and cytidine deaminase inhibitor

Orally active 5-LOX inhibitor

Selective 5-HT uptake inhibitor

Heme oxygenase and guanylyl cyclase inhibitor

Selective β₂ agonist

Cell-permeable inhibitor of atypical PKC isozyme PKMζ

Control peptide for ZIP (Cat. No. 2549)

Biotinylated peptide for ZIP (Cat No. 2549)

5-HT_2A/D₂ antagonist; atypical antipsychotic

Glutamate carboxypeptidase II and III (NAALADase, NAAG peptidase) inhibitor

Potent estrogen receptor antagonist

Competitive AMPA/kainate antagonist

Selective, non-peptide CCR8 agonist

Potent benzodiazepine agonist

Potent, competitive benzodiazepine antagonist

K_ATP channel opener

Potent, highly selective A_2A antagonist

Inhibitor of VEGF receptor tyrosine kinase

Potent, selective inhibitor of VEGFR-2

Potent, selective c-Raf inhibitor

Potent, selective JAK3 inhibitor

Inhibits Aurora kinase B

Potent, selective JAK3 inhibitor

Potent, centrally active H₂ antagonist

Benzodiazepine agonist

Selective NHE-1 inhibitor

Blocks voltage-sensitive Na⁺ and Ca²⁺ channels (T-type)

Benzodiazepine agonist