All Products

Cat.No.

Product Name / Activity

Antibody recognizing TRPV1 receptors

Highly potent, selective PDE5 inhibitor

Potent liver X receptor (LXR) agonist

GnRH receptor antagonist

Highly potent and selective PPARγ antagonist

Potent, orally active ghrelin receptor agonist

GABA_A agonist. Also GABA-T substrate and GABA uptake inhibitor

Cholinesterase inhibitor

Potent and selective ErbB2 inhibitor

Chloride channel blocker (hCLCA1/mCLCA3 and Cl^-/HCO₃^- exchange)

Synthetic thyrotropin-releasing hormone (TRH) analog

Estrogen receptor partial agonist/antagonist

Selective α_1A antagonist

Selective 5-HT_1A partial agonist

Non-selective, endogenous glycine receptor partial agonist

Selective PP1 inhibitor

Promotes assembly and inhibits disassembly of microtubules

α5-selective GABA_A inverse agonist

Selective cell-permeable CK2 inhibitor

Potent, selective non-transportable inhibitor of EAATs

High affinity σ₁ ligand

α7-selective agonist

Selective partial agonist at α4β2 receptors

Potent, high affinity 5-HT_2A agonist

Fragment 1-13 of GSK-3β sequence

Scrambled control peptide for use with TCS 183

Potent Chk1 inhibitor

Potent FLT3 inhibitor

Selective inhibitor of PTP1B

Orally active, subtype-selective NR1A/NR2B antagonist

Selective inhibitor of JNK2 and JNK3

Potent and selective OX₂ antagonist

Selective, ATP-competitive Pim-1 kinase inhibitor

Selective, ATP-competitive Pim kinase inhibitor

Antiprion agent; potently inhibits PrP-res accumulation

5-, 12-, 15-Lipoxygenase inhibitor

Potent CCR2b antagonist

Potent selective M₁ antagonist

DNA-methylating antitumor agent

Superoxide scavenger; antioxidant

NSAID, cyclooxygenase (COX-1) inhibitor. Also opener of K_IR2.3

Reverse transcriptase inhibitor

Activates p53 transcriptional activity

α₁ and α_2B antagonist (α₁ > α_2B). Orally active

Selective inhibitor of BTK

Potent, selective blocker of inward-rectifier K⁺ channels

Endogenous androgen receptor agonist

Potent inhibitor of vesicular monoamine transport; depletes dopamine stores

Non-selective K⁺ channel blocker

Cannabinoid receptor agonist; psychoactive

Highly potent NMDA receptor agonist

MAO-A inhibitor

Na⁺ channel blocker

Na⁺ channel blocker. Citrate salt of Cat. No. 1078

High affinity EAAT1 and EAAT2 blocker

PAR₁-activating peptide

TNF-α synthesis inhibitor

Potent inhibitor of SERCA ATPase

Potent subtype-selective ligand; ERα agonist/ERβ antagonist

Glutamate receptor ligand

Adenosine receptor antagonist; bronchodilator

Antibiotic. Inhibits vitronectin cell adhesion

H₃ antagonist and H₄ inverse agonist

Dopamine receptor antagonist; antipsychotic

Antibiotic, inhibits protein synthesis

Potent and selective P2Y₂ agonist

GABA_A agonist

Potent and selective MC₄ receptor agonist

Causes platelet aggregation and secretion

Potent actin polymerization regulator

Selective facilitator of 5-HT uptake; antidepressant

β₁ antagonist

Heme oxygenase inhibitor

Potent, selective H₂ antagonist

α₂ agonist

VGF-derived peptide

Neuronal nicotinic receptor antagonist

Cytochrome P450 1B1 inhibitor

Methionine aminopeptidase-2 inhibitor; antiangiogenic

Potent, selective P2X antagonist

Novel fluorescent cannabinoid ligand. Fluorescent form of AM 251

Compound library

80 kinase inhibitors supplied pre-dissolved in DMSO (250μl 10mM solutions)

1120 biologically active compounds pre-dissolved in DMSO (50μl 10mM solutions)

Compound library

1120 biologically active compounds pre-dissolved in DMSO (250μl 10mM solutions)

Water-soluble emulsion; negative control for Cat. Nos. 1017, 1685, 1686, 1781, 1782, 1783 and 2756

Potent, selective noradrenalin re-uptake inhibitor

GluR5 antagonist; anticonvulsant

Potent, selective inhibitor of IKK-2

Selective GABA_C antagonist

Subtype-selective GABA_A allosteric modulator

Highly selective IK_Ca1 channel blocker

Targets soluble Aβ to decrease amyloid plaque deposition. Also GABA analog

Antiallergic, inhibits release from mast cells

Potent and selective NOP antagonist

PAR₁ peptide fragment (residues 42-47); acts as a PAR₁ agonist

Ultrapotent inhibitor of PDE3

Histone deacetylase inhibitor

nNOS/iNOS inhibitor

Dihydrofolate reductase inhibitor

Standard H₁ antagonist, highly potent

Inhibits TNF-α-induced NF-κB activation

Potent, selective inhibitor of mitotic kinesin Eg5

Binds voltage-dependent anion channel (VDAC)

Selective PPARγ agonist; antidiabetic agent

5-HT₃ antagonist

Selective M₄ muscarinic antagonist

Potent 5-HT₃ receptor antagonist; orally active

Antibiotic; inhibits bacterial DNA synthesis

Blocking peptide for anti-TRPV1 (Cat. No. 2233)

Retinoic acid agonist

Nicotinic receptor antagonist

EGFR-kinase inhibitor

EGFR-kinase inhibitor