All Products

Cat.No.

Product Name / Activity

Antibody recognizing RacGAP

Diacylglycerol kinase inhibitor; increases PKC activity

Potent and selective B₁ antagonist

Potent and selective B₁ antagonist

Inhibitor of 14.3.3 proteins; induces apoptosis

TRPV1 antagonist peptide

Potent, selective 5-HT_2A antagonist

Control peptide version of Rac1 Inhibitor W56 (Cat. No. 2221)

Selective inhibitor of Rac1-GEF interaction

Potent, selective D₂/D₃ antagonist

Hsp90 inhibitor. Antifungal antibiotic

Selective estrogen receptor modulator (SERM)

Selective H₂ antagonist

Antianginal, activates pyruvate dehydrogenase

mTOR inhibitor; immunosuppressant

α₂ antagonist

Somatostatin analog

Potent, selective noradrenalin uptake inhibitor; orally active

Selective α_1B antagonist

NMDA antagonist; blocks ion channel and allosteric modulatory site

Selective D₂-like antagonist

K_ATP channel blocker

Inhibitor of vesicular monoamine transport

Ultrapotent vanilloid receptor agonist

Cyclooxygenase inhibitor

Endogenous retinoic acid receptor agonist. Also modulates PPARδ

Antitumor agent; suppresses mutant p53-bearing cancer cells

Selective MRP1 and P-gp inhibitor

Selective NPFF₁ and NPFF₂ antagonist

Non-nucleoside DNA methyltransferase inhibitor

Integrin binding sequence; inhibits integrin receptor function

Diacylglycerol lipase inhibitor

α₂ agonist. Also I₁ ligand

Glutamate release inhibitor/GABA uptake inhibitor

σ₂ antagonist. Also DAT inhibitor

Farnesyl diphosphate (FPP) synthase inhibitor

5-HT_2A antagonist

p53-MDM2 interaction inhibitor; antitumor

Potent 5-HT₂ antagonist

α4β2 selective nicotinic agonist

Nicotinic receptor agonist

Control peptide for TFLLR-NH₂ (Cat. No. 1464)

Selective TRPV4 antagonist

Selective TRPV4 agonist

Selective P2X₁ antagonist

Selective NR2B antagonist

Potent and selective 5-HT₆ antagonist

Inhibits NGF binding to p75^NTR and TrkA

Selective D₄ receptor partial agonist

Inhibitor of NF-κB activation

Benzodiazepine partial inverse agonist

Benzodiazepine inverse agonist

PDE4 inhibitor

Subtype-selective NR2B antagonist

Competitive inhibitor of IL-2/ IL-2Rα receptor interaction

Protein kinase inhibitor

Potent, orally active PKC inhibitor

Potent, collagenase-selective MMP inhibitor

Potent, selective 5-HT_2C agonist

Potent kynurenine 3-hydroxylase inhibitor

Selective NR2B antagonist

Inhibitor of Aβ42 fibril formation

Selective P2X₃ and P2X_2/3 antagonist

PDE4 inhibitor

PDE4 inhibitor. More active enantiomer of Cat. No. 0905

PDE4 inhibitor. Less active enantiomer of Cat. No. 0905

Selective D₂-like agonist

Potent H₃ antagonist

Anti-inflammatory, cytostatic and anti-viral

Inhibits complex I of the mitochondrial electron transport chain

Reported PKCδ inhibitor

Dopamine D₂ autoreceptor agonist. Also has affinity for D₃, D₄, 5-HT_1A receptors and the 5-HT transporter

Potent and selective NK₁ antagonist

Tyrosine kinase substrate peptide

Potent, subtype-selective α_1A antagonist

Selective 5-HT_2C antagonist

CCR2b chemokine receptor antagonist

Selective, high affinity 5-HT_2B antagonist

5-HT₃ ligand. Also shows affinity for zacopride binding site

α_1A antagonist

5-HT₄ antagonist

Potent PDE4 inhibitor

5-HT₄ antagonist

High affinity I₂ ligand. Highly selective

Highly selective CCR2 chemokine receptor antagonist

5-HT₃ partial agonist

5-HT₄ partial agonist

5-HT₄ partial agonist

Potent, selective α₂ antagonist

5-HT_1B/1A agonist

Mineralocorticoid receptor antagonist

Potent, selective mineralocorticoid receptor antagonist

Pure antiestrogen

Caged 4-aminopyridine; a non-selective K_V channel blocker

Caged GABA; excitable by visible wavelength

Caged Glutamate; excited by visible wavelengths

Prolongs inactivation of sodium channels; anticonvulsant

Non-selective Ca²⁺ channel blocker (N- and P-type)

Selective CB₁ agonist

Toll-like receptor 7 (TLR7) agonist

Potent, selective p38α and p38β inhibitor

Potent, selective α_2D antagonist

Ca²⁺ release inhibitor

Cyclin-dependent kinase 4 (cdk4) inhibitor

High affinity NOP ligand

Potent, selective NOP partial agonist peptide