All Products

Cat.No.

Product Name / Activity

Potent and selective sst₂ agonist

Potent, selective non-peptide NPY Y₅ antagonist

Selective EP₄ receptor antagonist

Potent PPARδ agonist

Potent, orally active human glucagon receptor antagonist

DNA ligase I, III and IV inhibitor

KCNQ1 (K_VLQT1) channel activator, activates I_Ks

Selective CCK₂ antagonist

Potent, non-peptide oxytocin receptor antagonist

Potent and selective oxytocin receptor antagonist

Ca²⁺ channel blocker

Potent, selective thromboxane A₂/prostaglandin endoperoxide antagonist

Selective for α5-containing GABA_A receptors

Potent, selective thromboxane A₂/prostaglandin endoperoxide antagonist

Potent and selective γ-secretase inhibitor

Very potent NMDA antagonist

Cell permeable prodrug of the IMPase inhibitor L-690,330 (Cat. No. 0681)

Inositol monophosphatase inhibitor

Potent, non-peptide ghrelin receptor agonist

High affinity σ ligand

5-HT_1D agonist

NMDA antagonist, acts glycine site

NMDA antagonist, acts glycine site

Selective 5-HT_1D receptor agonist

Potent, selective NK₁ antagonist

Potent NK₁ antagonist

Highly selective D₄ antagonist

High affinity D₂ antagonist

Highly selective D₄ antagonist

Selective β₃ antagonist

Very potent and selective β₃ partial agonist

Highly selective CB₂ agonist

High affinity, selective CB₂ agonist

Potent Raf kinase inhibitor

Potent and highly selective EP₃ antagonist

Substrate-competitive inhibitor of GSK-3

Potent and selective sst₄ agonist

Potent and selective sst₅ agonist

Subtype-selective GABA_A partial agonist

Cell-permeable, potent and selective proteasome inhibitor

Inhibits glutamate release. Anticonvulsant

Inhibits glutamate release. Water-soluble salt of Cat. No. 1611

H⁺,K⁺-ATPase inhibitor

Intermediate in lipid metabolism

EGFR, p60^c-src inhibitor

Selective MAO-B inhibitor

Dopamine precursor

Selective RARβ antagonist

Potent and selective dopamine D₁ antagonist

CB₁ agonist

Dihydroorotate dehydrogenase inhibitor

Fluorogenic caspase substrate

Cell-permeable caspase-9 inhibitor

Synthetic leptin peptide fragment

Inhibits nuclear export of proteins; antitumor

Ca²⁺ channel blocker (L-type)

JAK2, FLT3 and TrkA inhibitor

BLT₁/BLT₂ receptor agonist and potent chemotactic factor

Inhibits trypsin-like/cysteine proteases

GnRH receptor agonist

K_ATP channel opener. Active enantiomer of Cat. No. 1377

Antiepileptic; binds SV2A

Potent, selective BTK inhibitor

Blocks retinoic acid metabolism

Na⁺ channel blocker

Antibiotic; inhibits protein synthesis in gram-positive bacteria

Immunomodulator with antiangiogenic properties

KCNQ channel blocker

Amphibian bombesin-like peptide

Nicotinic agonist

Insect tachykinin-related peptide (TRP)

Broad spectrum cation channel blocker; neuroprotective

5-HT and noradrenalin re-uptake inhibitor (SNRI)

Mitochondrial hexokinase inhibitor

Peripherally acting μ agonist. Also Ca²⁺ channel blocker

Peripheral H₁ antagonist; antiallergic agent

Acts at the benzodiazepine modulatory site

Subtype-selective GABA_A receptor modulator

HMG-CoA reductase inhibitor

5-HT₇ agonist

High affinity 5-HT₇ agonist

Control peptide for SLIGRL-NH₂ (Cat. No. 1468)

Anti-inflammatory, antioxidant and free radical scavenger

Competitive melatonin MT₁/MT₂ antagonist

Selective, orally active LTD₄ antagonist

Novel, potent anandamide uptake inhibitor. Inhibits FAAH

Potent CCK₂ antagonist

Competitive NMDA receptor antagonist

Competitive NMDA antagonist

Potent and selective GlyT1 inhibitor

Selective, competitive BLT₂ receptor antagonist

High affinity 5-HT_2B antagonist, orally active

Selective CCK₂ antagonist

Selective PI 3-kinase inhibitor

Negative control of LY 294002 (Cat. No. 1130)

5-HT_1D-preferring antagonist

Selective CB₁ receptor antagonist/inverse agonist

Selective 5-HT_1F agonist

Highly potent, selective group II antagonist

Potent, selective 5-HT_1F agonist

Potent and highly selective group II mGlu agonist

Selective inhibitor of TGF-βRI

Selective mGlu_1a antagonist

Highly selective group II mGlu agonist

Dual 5-HT_1B/1D antagonist and 5-HT re-uptake inhibitor

Selective mGlu₁ antagonist

Positive allosteric modulator selective for mGlu₂

Inhibits Lyn-dependent activities of IL-5 receptor; cell-permeable

Pro-opiomelanocortin (POMC) derived peptide