All Products

Cat.No.

Product Name / Activity

Antibody recognizing GAL₁ (C' terminus)

Antibody recognizing GAL₁ (internal region)

Antibody recognizing GAL₂

Antibody recognizing GAL₃

Antibody recognizing K_IR3.2

Antibody recognizing rat GluR4 subunits

Antibody recognizing rat GluR5 subunits

Antibody recognizing rat GluR6 and GluR7 subunits

Antibody recognizing rat glutamate receptor δ1 and δ2 subunits

Antibody recognizing GLAST

Antibody recognizing GLT-1

Antibody recognizing GluR5

Antibody recognizing NR1 subunits

Antibody recognizing NR2B subunits

Antibody recognizing rat GluR1 subunits phosphorylated at Ser⁸³¹

Potent and highly selective GPR30 agonist

High affinity and selective GPR30 antagonist

Endogenous agonist

Anticonvulsant. Increases brain GABA

Serine protease inhibitor; inhibits thrombin, trypsin, kallikrein and plasmin

Non-selective galanin receptor agonist

Galanin receptor agonist

Galanin receptor agonist peptide

Endogenous galanin receptor agonist

Selective GAL₂ peptide agonist

Cholinesterase inhibitor

Inhibitor of βγ signaling

Selective, non-peptide GAL₁ agonist

Apoptosis inducer. Activates caspases and inhibits Bcl-2 family proteins

Potent, positive allosteric modulator of GABA_A receptors

Gap junction blocker; inhibits smooth muscle contraction and IP₃-mediated ATP release

Selective gap junction blocker

Selective CCK₂ agonist

Potent and selective glycine site antagonist. Orally available and active in vivo

High affinity benzodiazepine agonist

Potent, selective dopamine uptake inhibitor

Selective DA uptake inhibitor. Also σ ligand

Selective dopamine uptake inhibitor

Potent dopamine uptake inhibitor

Hsp90 inhibitor; anticancer and antimalarial activity

Selective Hsp90 inhibitor

DNA synthesis inhibitor

EGFR kinase inhibitor. Also estrogen and PPARγ ligand

Protein kinase C inhibitor

Endogenous ghrelin receptor agonist

Endogenous ghrelin receptor agonist

Major circulating form of ghrelin; devoid of activity at GHS receptor

Endogenous ghrelin receptor ligand

Major circulating form of ghrelin; devoid of activity at ghrelin receptor but is active in vivo

Ghrelin receptor antagonist

PAF receptor antagonist

Highly potent insulinotropic peptide

Potent insulinotropic gut hormone

Immunomodulator; reduces production of pro-inflammatory cytokines

K⁺ channel blocker (K_ATP)

K_ATP channel opener

Immunosuppressant; inhibits NF-κB and cytokine production

Metabolite of GLP-1-(7-36) (Cat No. 2082)

Endogenous hormone; displays intestinotrophic activity

Endogenous hormone; displays intestinotrophic activity

Glucagon receptor antagonist

Endogenous pancreatic peptide

Potent insulinotropic peptide

Blocking peptide for anti-GluR4 (Cat. No. 2046)

Blocking peptide for anti-GluR6/7 (Cat. No. 2048)

Blocking peptide for anti-glutamate receptor δ 1/2 (Cat. No. 2049)

Blocking peptide for anti-glutamate transporter GLAST (Cat. No. 2064)

Blocking peptide for anti-glutamate transporter GLT-1 (Cat. No. 2063)

Endogenous, non-selective agonist. Less active enantiomer

Endogenous, non-selective agonist

Endogenous potentiator, co-transmitter

Inhibits fibrin polymerization

NMDA receptor partial agonist; acts at the glycine site

Inhibitor of protein kinases G and A

Potent, selective κ antagonist

Selective κ/δ opioid heterodimer receptor agonist

Potent protein kinase C inhibitor; selective for α and β isozymes

Broad spectrum PKC inhibitor

GnRH receptor agonist

Pro-apoptotic; downregulates Bcl-2 and Bcl-XL

Highly selective CB₂ agonist

Selective CB₂ agonist

Inhibits G protein activation by GPCRs

Highly selective D₃ antagonist

Potent, selective 5-HT₄ antagonist

Potent, selective 5-HT₄ antagonist. Active in vivo

Potent, selective 5-HT_1B/1D antagonist

High affinity melatonin MT₃ ligand

Glycoprotein IIb/IIIa (α_IIbβ₃) receptor antagonist. Antithrombotic

Non-peptide, potent NK₂ antagonist

Potent NPY Y₁ antagonist/NPY Y₄ agonist. Binds to NPFF receptors

Potent thromboxane A₂/TP receptor antagonist

5-HT_1D agonist

5-HT_1B antagonist

Potent, selective NK₂ agonist

Potent, selective NK₁ agonist

A₁ agonist

Tachykinin NK₁ receptor antagonist

Subtype-selective κ opioid agonist

Potent, selective NK₂ antagonist

5-HT₃ antagonist

VIP antagonist

Stimulates growth hormone release

GRK2 inhibitory polypeptide. Gβγ antagonist

Selection of 5 group I mGlu receptor ligands (Cat. Nos. 0805, 0188, 1237, 1212 and 0337)

Selection of 5 group II mGlu receptor ligands (Cat. Nos. 1208, 0975, 1209, 0971 and 0337)

Selection of 5 group III mGlu receptor ligands (Cat. Nos. 0103, 1220, 0972, 0803 and 1209)

Endogenous GRP receptor agonist

Endogenous GRP receptor agonist

Positive modulator at GABA_B receptors

Selective PPARδ antagonist

Endothelial lipase and lipoprotein lipase inhibitor

Selective Rho-kinase (ROCK) inhibitor

Selective ERRγ and ERRβ agonist

Serum- and glucocorticoid-regulated kinase (SGK) inhibitor

Class III receptor tyrosine kinase (RTK) inhibitor

α₂ agonist. Also I₂ selective ligand

α_2A agonist

Endogenous activator of intestinal guanylyl cyclase

Broad spectrum steroid receptor ligand. Antagonizes FXR and displays hypolipidaemic activity

Broad spectrum steroid receptor ligand. More active isomer of Cat. No 2013

Specific GABA uptake inhibitor

Highly selective, potent PPARδ agonist

Selective PPARγ agonist. Orally active

Potent, selective human leukocyte elastase inhibitor

Orally active liver X receptor (LXR) agonist

Selective, high affinity CB₂ receptor partial agonist

Selective farnesoid X receptor (FXR) agonist

Potent, selective TrkA inhibitor

Potent, selective c-Raf1 kinase inhibitor

Potent dual EGFR/ErbB2 inhibitor; orally active

PPARα antagonist

Highly selective, potent PPARα agonist. Orally active

P2X₇ allosteric modulator

Selective inhibitor of PLK1 and PLK3

Potent and selective FFA1 (GPR40) agonist

Selective PPARγ antagonist

Non-competitive AMPA antagonist

Selective non-competitive AMPA antagonist