All Products

Cat.No.

Product Name / Activity

Antibody recognizing CB₂ receptors

Antibody recognizing CCK₁

Antibody recognizing mouse CCK₁

Antibody recognizing CCK₂

Antibody recognizing Cdk1 and Cdk2

Antibody recognizing Cdk2

Antibody recognizing c-Fos

Antibody recognizing c-Jun

Antibody recognizing CK1δ

Antibody recognizing CK1ε

Antibody recognizing COX-1

Antibody recognizing COX-2

Antibody recognizing CRF₁

Potent CCR4 antagonist

Protein kinase C inhibitor

Endogenous NK₁ agonist

Selective D₂-like agonist

Specific inhibitor of NF-κB activation

Phosphopeptide ligand for src SH2 domain

A₁ and A_2B antagonist. CNS stimulant

Selective calcineurin inhibitor

Vitamin D₃ analog

Affects bone formation and resorption

Vitamin D receptor (VDR) agonist

Commonly used laboratory reagent

Calmodulin antagonist

Cell-permeable calmodulin antagonist

Cell-permeable calmodulin agonist

Cell-permeable calmodulin agonist

Selective calpain inhibitor

Calpain and cathepsin L inhibitor

Potent, selective and photo-dependent PKC inhibitor

Protein phosphatase 1 and 2A inhibitor

Orally active protease inhibitor

DNA topoisomerase inhibitor

Calmodulin antagonist

NOS inhibitor

Natural cannabinoid; GPR55 antagonist, weak CB₁ antagonist, CB₂ inverse agonist and AMT inhibitor

Selection of 3 CB₁ receptor ligands (Cat. Nos. 1319, 1121 and 1117)

Mineralocorticoid receptor antagonist

Protein phosphatase 1 and 2A inhibitor

Prototypic vanilloid receptor agonist

Vanilloid receptor antagonist. Also activator of ENaCδ

Cholinergic receptor agonist

Gap junction blocker. Also inhibitor of 11 β-hydroxysteroid dehydrogenase

High affinity σ₁ ligand

Aromatic L-amino acid decarboxylase inhibitor

DNA cross-linking antitumor agent

5-HT₁ agonist. Also has high affinity for 5-ht_5A and 5-HT₇

Ionotropic glutamate receptor antagonist

Broad spectrum EAA ligand

Group I antagonist/group II agonist

Group I antagonist/group II agonist

Moderately potent NMDA antagonist

Broad spectrum EAA ligand

Competitive group I mGlu antagonist/weak group II agonist

Stable, water-soluble deactivator of NO

Highly selective H₃ antagonist

Selective, peripherally acting D₂-like agonist

Neuromodulating neuropeptide fragment; inhibits food intake in vivo

β-adrenoceptor and α₁-adrenoceptor antagonist

Glucosidases α and β inhibitor

Non-competitive nicotinic cholinergic antagonist

Potent dual CB₁/CB₂ agonist

High affinity, selective CB₂ agonist

Blocking peptide for Cat. No. 2231

Benzodiazepine inverse agonist, putative endogenous ligand

Oxidative phosphorylation uncoupler

Inhibitor of regulator of G-protein signaling 4 (RGS4)

Potent group II mGlu agonist

Potent, competitive glutamate uptake inhibitor

Non-sulfated form of CCK octapeptide

C-terminal octapeptide of CCK

Used to characterize NR2B-containing NMDA receptors

Hsp90 inhibitor

Potent and selective RARγ agonist

Selective RARβ/γ antagonist

RARγ-selective agonist

Positive allosteric modulator at mGlu₅

Neuroprotective; increases EAAT2 expression and activity

Antioxidant and anti-inflammatory

Selective COX-2 inhibitor

Ser/Thr protein phosphatase activator

Selective H₁ antagonist

Potent GnRH antagonist

Selective M₁ agonist

Soluble guanylyl cyclase (sGC) activator

Non-competitive AMPA antagonist

Blocking peptide for Anti-c-Fos (Cat. No. 2066)

Voltage-independent, selective CFTR chloride channel blocker

A₁, A_2B and A₃ antagonist and inhibitor of p38 MAPK and PDE4

Selective inhibitor of ATR and ATM kinases

Protein kinase G inhibitor

β₃ partial agonist. β₁/β₂ antagonist.

Positive modulator at GABA_B receptors

Highly potent and selective β₁ antagonist

Brain penetrant, selective GABA_B antagonist

Antagonist of mitochondrial Na⁺/Ca²⁺ exchange

Potent selective NMDA antagonist

Potent, selective and competitive NMDA antagonist

Selective, high affinity AT₂ ligand

Brain penetrant, selective GABA_B antagonist

Potent, selective GABA_B antagonist

Selective inhibitor of PKCβII

Potent, selective GABA_B antagonist

Potent, selective GABA_B antagonist

Selective inhibitor of Mnk1

Highly selective and potent non-peptide NPY Y₅ receptor antagonist

Potent, selective glycine-site NMDA antagonist

Positive modulator at GABA_B receptors

CGRP receptor agonist

Potent vasodilator

CGRP₁ receptor antagonist

CGRP₁ receptor antagonist

5-HT_1B agonist

Potent adenosine receptor antagonist

Potent, competitive NMDA antagonist

Selective central benzodiazepine receptor partial agonist

A_2A agonist

Endothelin-converting enzyme (ECE) inhibitor

Calmodulin antagonist

Potent retinoic acid receptor (RAR) agonist

Zwitterionic detergent

K⁺ channel blocker (high conductance, Ca²⁺-dependent)

Potent protein kinase C inhibitor

Potent inhibitor of L-glutamate uptake into synaptic vesicles

Nicotinic antagonist; slow offset

Potentiates GABA_A receptor function

Skeletal muscle relaxant

Adenosine receptor agonist

Sodium salt of Cat. No. 0237. Potent competitive inhibitor of L-glutamate uptake

Potent competitive inhibitor of L-glutamate uptake

Melatonin agonist

Potent, selective A₁ agonist

Tryptophan hydroxylase inhibitor

Potent and specific 5-HT₃ agonist

Urokinase inhibitor

Weak NMDA antagonist

mGlu₅ selective agonist

I_Ks blocker. Also blocks I_CFTR

I_Ks blocker. Enantiomer of (Cat. No. 1412)

Highly selective, orally active ET_A antagonist

Dihydrofolate reductase inhibitor

Selective inhibitor of GAT-1

Acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor

Potent and selective CCK₂ antagonist

Histone deacetylase inhibitor

Selective protein kinase D inhibitor

Selective PPARγ agonist

Dipeptidase inhibitor

Ca²⁺ channel blocker (dual L/N-type)

PDE3 inhibitor

PDE3A inhibitor. Also adenosine uptake inhibitor

β agonist

H₂ antagonist, I₁ agonist

Potent, selective CysLT₁ (LTD₄) antagonist; orally active

Selective 5-HT₂ antagonist

Selective α₁ agonist

5-HT₄ agonist; stimulates intestinal ACh release

Potent pro-apoptotic anticancer agent; activates caspase-3

Highly potent and selective 5-HT uptake inhibitor

Selective CAR agonist

Selective 5-HT₄ partial agonist

Peptide inhibitor of JNK/c-Jun interaction

Benzodiazepine agonist

Highly selective β₃ agonist

Selective inhibitor of MMP-13

H₁ antagonist

Subtype-selective AMPA agonist (GluR1 and GluR2)

Highly selective A₃ agonist

Highly potent H₃ antagonist and H₄ partial agonist

Deoxycytidine kinase (dCK) substrate

PPAR agonist

PPAR agonist

5-HT re-uptake inhibitor

α₂ agonist. Also I₁ ligand

Selective P2Y₁₂ antagonist

Water-soluble PGF_2α analog and potent FP receptor agonist

Dopamine antagonist with some D₄ selectivity. Also 5-HT_2A/2C antagonist

D₂-like antagonist. Displays some D₄ selectivity

Non-ATP-competitive p38α inhibitor

Potent AMPA/kainate antagonist

Potent AMPA/kainate antagonist. More water soluble form of Cat. No. 0190

Highly selective NR2B antagonist

State-dependent Na⁺ channel blocker; anticonvulsant

Inhibitor of monoamine transporters

Antioxidant

apoE peptide fragment

Inhibitor of tubulin

Inhibits tubulin polymerization. Antitumor, antiangiogenic and antimetastatic

Selective DNA-PK and mTOR inhibitor

γ-secretase inhibitor

C3-binding protein, inhibits complement activation

Control peptide for Compstatin (Cat. No. 2585)

Potent non-competitive NMDA receptor antagonist

Non-competitive NMDA receptor antagonist

H⁺-ATPase (vacuolar) inhibitor

Potent and selective H₃ receptor antagonist

Selective α3β4 nAChR antagonist

α1β1δγ selective nAChR antagonist

Ca²⁺ channel blocker (N-type)

α7 and α9 selective nAChR antagonist

Potent α3β2 and β3 subunit selective nicotinic antagonist

Ca²⁺ channel blocker (N, P and Q-type)

Selective antagonist of α6-containing nicotinic receptors

Selective α3β2 nAChR antagonist

RNA synthesis inhibitor

Endogenous glucocorticoid

Endogenous neuropeptide; binds sst₁ - sst₅ and GHS-R1a

Ghrelin receptor antagonist

Inhibitor of human telomerase activity

Major metabolite of nicotine

Selective, non-peptide CRF₁ antagonist

p53-stabilizing agent

Non-peptide, potent K_V1.3 channel blocker

Potent and selective CRF₁ antagonist

Selective, non-competitive AMPA antagonist

Broad spectrum MMP inhibitor

Potent CB₁ agonist

Potent, non-selective cannabinoid receptor agonist

Selective PDE4 inhibitor

Potent and selective 5-HT_2C agonist

5-HT_1B agonist

Potent, selective 5-HT_1B agonist

Potent and selective NK₁ antagonist

Selective non-competitive mGlu₁ receptor antagonist

Dopamine uptake inhibitor

Potent NMDA antagonist. More active enantiomer of (RS)-CPP (Cat. No. 0173)

Potent NMDA antagonist

5-HT_2B/2C receptor agonist

Potent, competitive NMDA antagonist

Very potent group III mGlu antagonist

DNA topoisomerase I inhibitor; antitumor

Selective Epac activator

Subtype-selective weakly desensitizing AMPA agonist

CRF-binding protein inhibitor

Stimulates ACTH release

CRF receptor antagonist

K_ATP channel opener

Endogenous central CT receptor agonist

STAT3 inhibitor. Also displays multiple other activities

Selective and potent μ antagonist

Highly selective, potent μ antagonist

Endogenous peptide agonist at NPR2

Selective inhibitor of STAT3/JAK2 signaling

Antitumor, anti-inflammatory and antioxidant

Non-selective adenosine A₂ receptor agonist

AMPA receptor potentiator

Selective D₁-like agonist

5-HT_1A/1B antagonist. Also β-adrenergic antagonist

Selective, ATP-competitive PLK1 inhibitor

Inhibitor of protein synthesis

Inhibitor of hedgehog (Hh) signaling

Potent, selective A₁ agonist

Inhibitor of SERCA ATPase

Non-selective sst receptor antagonist

Calcineurin inhibitor

AMPA selective desensitization inhibitor

Selective sst₂ antagonist

Calcineurin inhibitor (protein phosphatase 2B)

Activator of SK2 and SK3 channels

Selective μ antagonist

5-HT₂ antagonist

NMDA and mGlu agonist

Potent, selective neuronal nicotinic agonist

Disrupts actin filament function