All Products

Cat.No.

Product Name / Activity

Selective GSK-3 phosphopeptide substrate

Promotes inclusion formation in Huntington's and Parkinson's diseases

Selective GABA_B agonist. Active enantiomer of (RS)-Baclofen (Cat. No. 0417)

Selective GABA_B agonist

PPARγ antagonist

H⁺-ATPase (vacuolar) inhibitor

Dual PI 3-kinase and PDK1 inhibitor

5- and 12-Lipoxygenase inhibitor

Selective agonist for the sensory neuron specific receptor (SNSR)

Opioid receptor agonist. Also agonist at the sensory neuron specific receptor (SNSR)

Selective Bax activator; induces Bax-mediated apoptosis

Potent and selective NOP antagonist

Prodrug topoisomerase II inhibitor

Selective calcium chelator

Cell-permeable Ca²⁺ chelator

Potent, broad spectrum MMP inhibitor

Inhibits Bax-mediated mitochondrial cytochrome c release

Inhibitor of Bax-mediated apoptosis

Inhibitor of Bax-mediated apoptosis

Negative control peptide for Bax inhibitor peptides V5 and P5 (Cat. Nos. 1785 and 1786)

Irreversible inhibitor of TNF-α-induced IκBα phosphorylation

Irreversible inhibitor of TNF-α-induced IκBα phosphorylation

Non-competitive mGlu₁ antagonist with inverse agonist activity

Soluble guanylyl cyclase (sGC) activator

Potent and selective VPAC₂ agonist

CB₁/CB₂ receptor partial agonist

Potent A_2B receptor agonist; cardioprotective

Ca²⁺-channel activator (L-type)

Ca²⁺-channel blocker (L-type)

Ca²⁺-channel activator (L-type)

Orally active 5-lipoxygenase activating protein (FLAP) inhibitor

Dual TP/DP₂ (CRTH2) receptor antagonist

Dual CysLT₁ and CysLT₂ antagonist

Selective urokinase (uPA) inhibitor

Selective PDE11 inhibitor

pH indicator

Modulates AMPA-mediated responses

TRPV1 antagonist

Potent, selective σ ligand

σ₁ selective antagonist

Selective σ₁ ligand, putative antagonist

Potent P2X₄ receptor antagonist

Activates TrkB and p75 receptors

γ-secretase inhibitor; lowers Aβ40 and Aβ42 levels

Angiotensin-converting enzyme (ACE) inhibitor

Cytostatic agent; exhibits DNA alkylating and purine analog properties

Calcium channel blocker

NCX inhibitor, Deg/ENaC channel blocker; amiloride (Cat. No. 0890) derivative

Nicotinic antagonist

δ₂ selective non-peptide antagonist

Non-selective calcium channel blocker

Aminopeptidase inhibitor

Selection of 3 β-adrenoceptor agonists (Cat. Nos. 0948, 1747 and 1660)

Selection of 3 β-adrenoceptor antagonists (Cat. Nos. 1024, 0821 and 1511)

Selective β₁ antagonist

Antitumor and anti-HIV agent; activates NF-κB. Also TGR5 agonist

H₃ receptor inverse agonist/antagonist

Potent, selective I₂ ligand. Putative agonist

High affinity 5-HT₆ antagonist

Potent, selective GABA_B positive allosteric modulator

Inhibitor of SERCA ATPase

D₂ receptor agonist. Also α₂ agonist and 5-HT₃ antagonist

Selective α2 agonist

Hepatocyte nuclear factor 4α (HNF4α) antagonist

Selective, competitive JNK inhibitor

Potent and selective CGRP receptor antagonist

Highly selective NPY Y₁ receptor antagonist

Mixed NPY Y₁ and NPFF receptor antagonist

Selective telomerase inhibitor

Selective inhibitor of EGFR-kinase

Highly selective EGFR-kinase inhibitor

Non-steroidal androgen receptor antagonist

Noradrenalin, 5-HT and dopamine re-uptake inhibitor

Water-soluble GABA_A antagonist

Water-soluble GABA_A antagonist

Water-soluble GABA_A antagonist

Potent GABA_A antagonist

MAO-A and MAO-B inhibitor

Selective Hsp90 inhibitor

Potent, selective non-peptide NPY Y₂ receptor antagonist

Bombesin/GRP receptor agonist

Bombesin antagonist

Selective neuromedin B receptor antagonist (NMB-R, BB₁)

sst₅ agonist

Somatostatin receptor ligand

NMB receptor antagonist. Also U-II receptor antagonist

Potent 5-HT₄ receptor full agonist

Selective positive allosteric modulator of mGlu₂

Standard κ selective antagonist

Potent, selective GSK-3 inhibitor

Selective α₄β₁ (VLA-4) inhibitor

Selective GSK-3α/β inhibitor

Versatile marker for neuroanatomical investigations

Bim peptide fragment

Muscarinic receptor antagonist; some selectivity for M₁

Potent dopamine uptake inhibitor

Potent PKC inhibitor and nicotinic receptor antagonist

β₁ antagonist

G9a-like protein and G9a histone lysine methyltransferase inhibitor

Putative K_2P2.1 (TREK-1) channel opener

Selective inhibitor of myosin II ATPase activity. Active enantiomer of (±)-blebbistatin (Cat. No. 1760)

Selective inhibitor of myosin II ATPase activity. Inactive enantiomer of (±)-blebbistatin (Cat. No. 1760)

Selective inhibitor of myosin II ATPase activity

Neurotoxic amino acid

Potent, selective CB₂ ligand

Highly selective, orally active non-peptide ET_A antagonist

Potent BK_Ca (K_Ca1.1) channel opener

Potent, competitive NPY Y₁ receptor antagonist

Selective RARα antagonist

Potent γ-secretase inhibitor

ATP citrate lyase inhibitor; orally bioavailable

Synthetic retinoid. RARβ agonist; also RARα and RARγ antagonist

Potent, selective MC₁ receptor agonist

Pan-RAR inverse agonist

Dual IR/IGF1R inhibitor

RARα-selective agonist

Selective RARγ agonist

High affinity, potent CCR2 antagonist

Sigma antagonist. Antipsychotic agent

Non-prostanoid prostacyclin IP receptor partial agonist

Selective α_1D antagonist

Standard δ₁ selective antagonist

FPR1 antagonist

Involved in gastrointestinal tract function

Bombesin receptor antagonist

Bombesin receptor antagonist

Potent bradykinin receptor agonist

Bioactive, bradykinin-related peptide

Antiangiogenic; inhibits threonyl-tRNA synthetase

Dual Src-Abl inhibitor; antiproliferative

Selective 5-HT_1A agonist

Orthosteric nAChR antagonist

Non-competitive GC inhibitor. Also AC inhibitor

Selective ET_B antagonist

Selective ET_A antagonist

Selective ET_B agonist

Endogenous agonist at bradykinin receptors (B₂ > B₁)

Potent and selective B₁ agonist

Bradykinin receptor agonist (B₁ > B₂)

Selective B₂ agonist

Potent bradykinin receptor agonist (B₂ > B₁)

Selective B₁ agonist

Endogenous peptide agonist at ANP receptor A (NRP1)

p90 ribosomal S6 kinase inhibitor

Disrupts protein translocation to Golgi

Benzodiazepine partial agonist

Selective h5-HT_1D antagonist

β₃ agonist

Selective α_2A antagonist

Selective PDE7 inhibitor

Potent and selective κ agonist

Potent 5-ht_1E/F agonist

Cell-permeable cAMP analog

cGMP analog; activates PKG

Selective D₂-like agonist

Potent agonist of α4β4, α4β2 and α7 nACh receptors

Selective nNOS inhibitor

Immunomodulatory and antitumor compound

Protein kinase C activator

Potent dopamine uptake inhibitor

Selective inhibitor of skeletal muscle myosin II ATPase activity

Potent SNRI; active metabolite of sibutramine (Cat. No. 2290)

MIF binder

Potent, selective I₂ ligand. Putative antagonist

Potent, highly selective I₂ ligand

Potent, highly selective I₂ ligand

β₁ and β₂ antagonist

Synthetic glucocorticoid; anti-inflammatory and chemopreventive

Na⁺/2Cl^-/K⁺ (NKCC) cotransporter inhibitor

α7 subtype-selective nAChR antagonist

Opioid receptor ligand

Non-selective inhibitor of dopamine and noradrenalin transporters

Mixed H₂/H₃ antagonist

5-HT_1A partial agonist

CCK-inactivating serine protease inhibitor

Highly selective NPY Y₁ receptor antagonist; devoid of Y₄ agonist activity

Non-competitive protein tyrosine phosphatase inhibitor; enhances insulin signaling

Potent, selective non-peptide δ agonist

5-HT_2B agonist

5-Lipoxygenase inhibitor

Highly selective NPY Y₅ agonist

Potent, selective CCR1 antagonist

Selective CCR1 antagonist

PDK1 inhibitor

Potent and selective inhibitor of iNOS

Selective PARP-1 inhibitor

PARP-1 and PARP-2 inhibitor

P2X₇ agonist. Also P2X₁ and P2Y₁ partial agonist