All Products

Cat.No.

Product Name / Activity

Antibody recognizing Bcl-2

Selective GSK-3 phosphopeptide substrate

Promotes inclusion formation in Huntington's and Parkinson's diseases

Selective GABA_B agonist. Active enantiomer of Cat. No. 0417

Selective GABA_B agonist

PPARγ antagonist

H⁺-ATPase (vacuolar) inhibitor

Dual PI 3-kinase and PDK1 inhibitor

5- and 12-Lipoxygenase inhibitor

Selective agonist for the sensory neuron specific receptor (SNSR)

Opioid receptor agonist. Also agonist at the sensory neuron specific receptor (SNSR)

Selective calcium chelator

Cell-permeable Ca²⁺ chelator

Potent, broad spectrum MMP inhibitor

Voltage-gated Na⁺ channel activator

Inhibits Bax-mediated mitochondrial cytochrome c release

Inhibitor of Bax-mediated apoptosis

Inhibitor of Bax-mediated apoptosis

Negative control peptide for Cat. Nos. 1785 and 1786

Irreversible inhibitor of TNF-α-induced IκBα phosphorylation

Irreversible inhibitor of TNF-α-induced IκBα phosphorylation

Non-competitive mGlu₁ antagonist with inverse agonist activity

Potent and selective VPAC₂ agonist

CB₁/CB₂ receptor partial agonist

Ca²⁺-channel activator (L-type)

Ca²⁺-channel blocker (L-type)

Ca²⁺-channel activator (L-type)

Dual TP/DP₂ (CRTH2) receptor antagonist

Dual CysLT₁ and CysLT₂ antagonist

pH indicator

Modulates AMPA-mediated responses

Potent, selective σ ligand

σ₁ selective antagonist

Selective σ₁ ligand, putative antagonist

Activates TrkB and p75 receptors

Angiotensin-converting enzyme (ACE) inhibitor

Cytostatic agent; exhibits DNA alkylating and purine analog properties

Nicotinic antagonist

δ₂ selective non-peptide antagonist

Aminopeptidase inhibitor

Selection of 3 β-adrenoceptor agonists (Cat. Nos. 0948, 1747 and 1660)

Selection of 3 β-adrenoceptor antagonists (Cat. Nos. 1024, 0821 and 1511)

Selective β₁ antagonist

Potent, selective I₂ ligand. Putative agonist

Potent, selective GABA_B positive allosteric modulator

Inhibitor of SERCA ATPase

D₂ receptor agonist. Also α₂ agonist and 5-HT₃ antagonist

Selective, competitive JNK inhibitor

Highly selective NPY Y₁ receptor antagonist

Mixed NPY Y₁ and NPFF receptor antagonist

Selective telomerase inhibitor

Selective inhibitor of EGFR-kinase

Highly selective EGFR-kinase inhibitor

Non-steroidal androgen receptor antagonist

Water-soluble GABA_A antagonist

Water-soluble GABA_A antagonist

Water-soluble GABA_A antagonist

Potent GABA_A antagonist

MAO-A and MAO-B inhibitor

Potent, selective non-peptide NPY Y₂ antagonist

Bombesin/GRP receptor agonist

Bombesin antagonist

Selective neuromedin B receptor antagonist (NMB-R, BB₁)

sst₅ agonist

Somatostatin receptor agonist

NMB receptor antagonist. Also U-II receptor antagonist

Standard κ selective antagonist

Potent, selective GSK-3 inhibitor

Versatile marker for neuroanatomical investigations

Bim peptide fragment

Muscarinic receptor antagonist; some selectivity for M₁

Potent dopamine uptake inhibitor

β₁ antagonist

G9a-like protein and G9a histone lysine methyltransferase (HMTase) inhibitor

Selective inhibitor of myosin II. Active enantiomer of Cat. No. 1760

Selective inhibitor of myosin II. Inactive enantiomer of Cat. No. 1760

Selective inhibitor of myosin II

Neurotoxic amino acid

Potent, selective CB₂ ligand

Highly selective, orally active non-peptide ET_A antagonist

Potent Maxi-K channel opener (BK_Ca, K_Ca1.1)

Potent, competitive NPY Y₁ antagonist

High affinity, potent CCR2 antagonist

Sigma antagonist. Antipsychotic agent

Non-prostanoid prostacyclin IP receptor partial agonist

Selective α_1D antagonist

Standard δ₁ selective antagonist

Involved in gastrointestinal tract function

Bombesin receptor antagonist

Bombesin receptor antagonist

Potent bradykinin receptor agonist

Bioactive, bradykinin-related peptide

Selective 5-HT_1A agonist

Non-competitive GC inhibitor. Also AC inhibitor

Selective ET_B antagonist

Selective ET_A antagonist

Selective ET_B agonist

Endogenous agonist at bradykinin receptors (B₂ > B₁)

Potent and selective B₁ agonist

Bradykinin receptor agonist (B₁ > B₂)

Selective B₂ agonist

Potent bradykinin receptor agonist (B₂ > B₁)

Selective B₁ agonist

Endogenous peptide agonist at ANP receptor A (NRP1)

Disrupts protein translocation to Golgi

Benzodiazepine partial agonist

Selective h5-HT_1D antagonist

β₃ agonist

Selective α_2A antagonist

Selective PDE7 inhibitor

Potent and selective κ agonist

Potent 5-ht_1E/F agonist

Cell-permeable cAMP analog

cGMP analog; activates PKG

Selective D₂-like agonist

Selective nNOS inhibitor

Protein kinase C activator

Potent dopamine uptake inhibitor

Selective inhibitor of skeletal muscle myosin II ATPase activity

Potent SNRI; active metabolite of sibutramine (Cat. No. 2290)

Potent, selective I₂ ligand. Putative antagonist

Potent, highly selective I₂ ligand

Potent, highly selective I₂ ligand

β₁ and β₂ antagonist

Synthetic glucocorticoid; anti-inflammatory and chemopreventive

Na⁺/2Cl^-/K⁺ (NKCC) cotransporter inhibitor

α7 subtype-selective nAChR antagonist

Opioid receptor ligand

Non-selective inhibitor of dopamine and noradrenalin transporters

Mixed H₂/H₃ antagonist

5-HT_1A partial agonist

CCK-inactivating serine protease inhibitor

Highly selective Y₁ antagonist; devoid of Y₄ agonist activity

Non-competitive protein tyrosine phosphatase inhibitor; enhances insulin signaling

Potent, selective non-peptide δ agonist

5-HT_2B agonist

5-Lipoxygenase inhibitor

Highly selective Y₅ agonist

Selective CCR1 antagonist

Potent and selective inhibitor of iNOS

P2X₇ agonist. Also P2X₁ and P2Y₁ partial agonist