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Displaying products alphabetically by name (A)

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Cat.No.
Product Name / Activity
2524A 205804

Selective inhibitor of E-selectin and ICAM-1 expression

2753A 350619 hydrochloride

Soluble guanylyl cyclase (sGC) activator

2972A 438079 hydrochloride

Competitve P2X7 antagonist

1052A 61603 hydrobromide

α1A agonist

1534A 68930 hydrochloride

Potent, selective D1-like agonist

3701A 740003

Potent and selective P2X7 antagonist

3336A 769662

Potent AMPK activator

1701A 77636 hydrochloride

Potent, selective D1-like agonist. Orally active

2976A 803467

Selective NaV1.8 blocker

2341A 80426 mesylate

High affinity α2 antagonist. Also 5-HT uptake inhibitor

2939A 83-01

Selective inhibitor of TGF-βRI, ALK4 and ALK7

3060A 841720

Selective mGlu1 antagonist

1234A23187, free acid

Calcium ionophore

0378A-7 hydrochloride

Calmodulin antagonist

2411A-71623

Potent and selective CCK1 agonist. Suppresses feeding

3025AA 2414

Thromboxane A2 (TP) receptor antagonist

1462AACOCF3

Phospholipase A2 inhibitor

151517-AAG

Selective Hsp90 inhibitor

1297Abn-CBD

Selective GPR55 agonist; neurobehaviorally inactive

2721ABS 205

Upregulates NCAM expression. Valproic acid (Cat No. 2815) derivative

2372ABT 702 dihydrochloride

Adenosine kinase inhibitor; orally active

2214ABT 724 trihydrochloride

Potent, selective D4 partial agonist; proerectile

3419AC 187

Potent and selective amylin receptor antagonist

3043AC 45594

SF-1 inverse agonist

3369AC 55541

Potent and selective PAR2 agonist

2436AC 55649

Selective RARβ2 agonist

2484(±)-AC 7954 hydrochloride

Non-peptide UT receptor agonist

09639-AC

Chloride transport inhibitor

1846Ac2-12

Annexin/lipocortin 1-mimetic; inhibits leukocyte extravasation

1845Ac2-26

Annexin/lipocortin 1-mimetic; inhibits leukocyte extravasation

3231Ac9-25

Annexin I N-terminal peptide. Acts as a FPR1 ligand

3618Acamprosate calcium

GABA agonist and glutamatergic modulator

2673Acarbose

Glucosidase α inhibitor (intestinal)

0258ACBC

NMDA antagonist, acts glycine site

0271cis-ACBD

Potent, selective L-glutamate uptake inhibitor

0270trans-ACBD

Selective, very potent NMDA agonist

2254ACDPP hydrochloride

Selective mGlu5 receptor antagonist

1319ACEA

Potent, highly selective CB1 agonist

3069Acephate

Anticholinesterase insecticide

2728ACET

Potent antagonist of GluR5-containing kainate receptors

1706Acetaminophen

Cyclooxygenase inhibitor; may be selective for COX-3

0722N-Acetyl-N-acetoxy-4-chlorobenzenesulfonamide

Nitroxyl precursor

0355(±)-Acetylcarnitine chloride

Intermediate in lipid metabolism

2809Acetylcholine chloride

Endogenous neurotransmitter

03524-Acetyl-1,1-dimethylpiperazinium iodide

Nicotinic agonist

0395N-Acetylglycyl-D-glutamic acid

Potent convulsant

0384N-Acetyl-L-leucyl-L-leucyl-L-methional

Cathepsin inhibitor

03511-Acetyl-4-methylpiperazine hydrochloride

Nicotinic agonist

1930N-Acetyl-O-phosphono-Tyr-Glu Dipentylamide

Phosphopeptide ligand for src SH2 domain

1927N-Acetyl-O-phosphono-Tyr-Glu-Glu-Ile-Glu

Phosphopeptide ligand for src SH2 domain

0357N-Acetyltryptamine

Melatonin partial agonist (MT1/MT2). Also MT3 antagonist

1762Acifran

Hypolipidaemic agent; agonist for the GPR109A (HM74A) and GPR109B receptors

2784Acipimox

Antilipolytic agent

1318ACPA

Potent, selective CB1 agonist

1781ACPA (in TocrisolveTM 100)

Potent, selective CB1 agonist (in water-soluble emulsion)

0284(1S,3R)-ACPD

Group I/group II mGlu agonist

0186cis-ACPD

Potent NMDA agonist. Also group II mGluR agonist

0187(±)-trans-ACPD

Group I/group II mGlu agonist

1111ACPT-I

Group III mGlu agonist

1112ACPT-II

Competitive mGlu receptor antagonist

3525ACSF

Artificial cerebrospinal fluid

3492ACTH (1-39)

Potent endogenous MC2 agonist

1229Actinomycin D

Inhibits RNA polymerase

3205ACV 1

α9α10-selective antagonist

2513Acyclovir

Inhibits viral DNA polymerase; antiherpetic agent

0860tADA

Group I agonist; some mGlu5 selectivity

2852Adapalene

RARβ and RARγ agonist

3716Adaphostin

p210bcr/abl kinase inhibitor

3624Adenosine

Endogenous adenosine receptor agonist

2651AEG 3482

Inhibitor of JNK signaling

1793AF 12198

Potent, selective human type I IL-1 receptor antagonist

1105AF-DX 116

Selective M2 antagonist

1345AF-DX 384

Potent M2/M4 antagonist

2730AG 045572

Selective GnRH receptor antagonist

1276AG 1478 hydrochloride

Highly potent EGFR-kinase inhibitor

0493AG 18

EGFR/PDGFR-kinase inhibitor

0503AG 213

EGFR/PDGFR-kinase inhibitor

0414AG 490

EGFR-kinase inhibitor. Also JAK2, JAK3 inhibitor

0619AG 494

Potent EGFR-kinase inhibitor

0618AG 555

Potent EGFR-kinase inhibitor

0616AG 556

EGFR-kinase inhibitor

1555AG 825

Selective ErbB2 inhibitor

0497AG 99

EGFR-kinase inhibitor

2799ω-Agatoxin IVA

Ca2+ channel blocker (P-type)

2802ω-Agatoxin TK

Ca2+ channel blocker (P/Q-type)

3233AGK 2

Selective SIRT2 inhibitor

0842Agmatine sulfate

α2 ligand. Also imidazoline ligand

1072AGN 192403 hydrochloride

I1 selective ligand

0998AH 11110 hydrochloride

Subtype-selective α1B ligand

0671AH 6809

EP1 and EP2 receptor antagonist

2840AICAR

AMPK activator

0904AIDA

Potent, selective group I mGlu antagonist

0678(+)-AJ 76 hydrochloride

Antagonist; preferential action at D2-like autoreceptors

1353Akt/SKG Substrate Peptide

Akt/PKB substrate (synthetic)

2422AKTide-2T

Akt/PKB substrate (synthetic)

0206β-Alanine

Endogenous glycine agonist, more selective than Taurine (Cat. No. 0209)

0204D-Alanine

Weak glycine receptor agonist

0205L-Alanine

Glycine receptor agonist, more potent than D-isomer (Cat. No. 0204)

3305Alfuzosin hydrochloride

Uroselective α1 antagonist

3653Allopregnanolone

GABAA receptor positive allosteric modulator

1871α1-Adrenoceptor TocrisetTM

Selection of 5 α1-adrenoceptor ligands (Cat. Nos. 1052, 0888, 1006, 0946 and 0623)

1872α2-Adrenoceptor TocrisetTM

Selection of 5 α2-adrenoceptor ligands (Cat. Nos. 1030, 0425, 0928, 1133 and 0891)

3046Alphaxalone

Direct activator and potentiator of GABAA

2806Alprenolol hydrochloride

β antagonist

1620Alprostadil

Prostaglandin. Vasodilator and antiplatelet agent in vivo

0485Alrestatin

Aldose reductase inhibitor

1809Altanserin hydrochloride

5-HT2A receptor antagonist

1757ALX 5407 hydrochloride

Selective non-transportable GlyT1 inhibitor

1893Alytesin

Amphibian bombesin-like peptide

2564AM 114

20S proteasome inhibitor

3381AM 1172

Anandamide uptake inhibitor. Also FAAH inhibitor and CB receptor partial agonist

1117AM 251

Potent CB1 antagonist. Also GPR55 agonist

1115AM 281

Potent, selective CB1 antagonist/inverse agonist

1116AM 404

Anandamide transport inhibitor

1685AM 404 (in TocrisolveTM 100)

Anandamide transport inhibitor (in water-soluble emulsion)

0760AM 580

Retinoic acid agonist

1120AM 630

CB2 selective antagonist/inverse agonist

3507AM 80

RARα agonist; anticancer

0876AM 92016 hydrochloride

KV channel blocker

0388Ambenonium dichloride

Cholinesterase inhibitor

2404Ambroxol hydrochloride

Na+ channel blocker

3299AMD 3100 octahydrochloride

Highly selective CXCR4 antagonist

2316AMG 9810

Potent and selective, competitive antagonist of TRPV1

0524AMI-193

D2-like receptor antagonist

0890Amiloride hydrochloride

Na+ channel blocker. Also I2 imidazoline ligand

07883-Aminobenzamide

PARP inhibitor

0787Aminoguanidine hydrochloride

Irreversible iNOS inhibitor

0721Aminopotentidine

H2 antagonist

2072Aminopurvalanol A

Cyclin-dependent kinase inhibitor

09404-Aminopyridine

Non-selective KV channel blocker

2132Amisulpride

Selective D2/D3 receptor antagonist; atypical antipsychotic agent

2571Amlodipine besylate

Ca2+ channel blocker (L-type)

2385AMN 082 dihydrochloride

The first selective mGlu7 agonist

1074(RS)-AMPA hydrobromide

Selective AMPA agonist. More water soluble form of (RS)-AMPA (Cat. No. 0169)

1822AMPA Receptor TocrisetTM

Selection of 5 AMPA receptor ligands (Cat. Nos. 0254, 0306, 1044, 0713 and 1454)

0253(R)-AMPA

Inactive isomer of (RS)-AMPA (Cat. No. 0169)

0169(RS)-AMPA

Selective AMPA agonist

0254(S)-AMPA

Selective AMPA agonist. Active isomer of (RS)-AMPA (Cat. No. 0169)

2746Amperozide hydrochloride

Atypical antipsychotic; high affinity 5-HT2 ligand

2813D-Amphetamine sulfate

Induces dopamine, 5-HT and noradrenalin release

1337cAMPS-Rp, triethylammonium salt

cAMP antagonist

1333cAMPS-Sp, triethylammonium salt

Cell-permeable cAMP analog

0871AMT hydrochloride

Potent, selective iNOS inhibitor

0668Amthamine dihydrobromide

Highly selective standard H2 agonist

3418Amylin

Endogenous peptide agonist for amylin, calcitonin, CGRP and adrenomedullin receptors

3391Amyloid β-peptide (42-1) (human)

Inactive control peptide for Cat. No. 1428

1892Amyloid β-Peptide (10-20) (human)

Amyloid β-peptide; substrate for MMP-2

1894Amyloid β-Peptide (12-28) (human)

Amyloid β-peptide; minimum required for binding to brain proteins

1191Amyloid β-Peptide (1-40) (human)

Amyloid β-protein fragment

2424Amyloid β-peptide (1-40) (rat)

Amyloid β-protein fragment

1428Amyloid β-Peptide (1-42) (human)

Predominant amyloid β-protein fragment

2425Amyloid β-peptide (1-42) (rat)

Predominant amyloid β-protein fragment

1938Amyloid β-Peptide (1-43) (human)

Amyloid β-protein fragment

1429Amyloid β-peptide (25-35) (human)

Human amyloid β-protein fragment functionally required for neurotoxicity

1971(+)-Anabasine hydrochloride

Neuronal nicotinic receptor agonist

2432Anagrelide hydrochloride

Potent PDE3 inhibitor

1339Anandamide

Endogenous CB receptor agonist

1017Anandamide (in TocrisolveTM 100)

Endogenous CB receptor agonist (in water-soluble emulsion)

3717Anandamide-d4

Deuterated anandamide. Endogenous CB receptor agonist

3388Anastrozole

Potent aromatase (CYP19) inhibitor

0789(±)-Anatoxin A fumarate

Nicotinic agonist

1562Angiotensin (1-7)

Vasorelaxant peptide

1563Angiotensin I (human, mouse, rat)

Endogenous precursor to angiotensin II (Cat. No. 1158)

1158Angiotensin II

Potent vasoconstrictor peptide

1564Angiotensin III (human, mouse)

Vasoconstrictor peptide

1897Angiotensin IV (human)

Agonist for the putative AT4 receptor

0867Aniracetam

Desensitization inhibitor (AMPA > kainate)

1290Anisomycin

Protein synthesis inhibitor

0703Anpirtoline hydrochloride

Highly potent 5-HT1B agonist. Also 5-HT3 antagonist

1954Antagonist G

Broad spectrum neuropeptide receptor antagonist

2778Antalarmin hydrochloride

CRF1 antagonist

0791Antazoline hydrochloride

Imidazoline ligand

3451Anti-AChE

Antibody recognizing AChE

3452Anti-ADRB1

Antibody recognizing β1 adrenoceptors

3450Anti-ADRB2

Antibody recognizing β2 adrenoceptors

3453Anti-AT1

Antibody recognizing AT1

3454Anti-Aurora A

Antibody recognizing Aurora A

2071Antisauvagine-30

Potent, selective and competitive CRF2 antagonist

3296AP 18

Reversible TRPA1 channel blocker

0125DL-AP3

Group I mGlu antagonist

3699DL-AP4 Sodium salt

Broad spectrum EAA antagonist

0102D-AP4

Broad spectrum EAA antagonist

0101DL-AP4

Broad spectrum EAA antagonist

0103L-AP4

Selective group III mGlu agonist

0106D-AP5

Potent, selective NMDA antagonist. More active form of DL-AP5 (Cat. No. 0105)

0105DL-AP5

Potent, selective NMDA antagonist

0107L-AP5

Potent, selective NMDA antagonist. Less active form of DL-AP5 (Cat. No. 0105)

0341L-AP6

Selective agonist of the 'quis' effect

0164D-AP7

Specific NMDA antagonist. More active form of DL-AP7 (Cat. No. 0104)

0104DL-AP7

Specific NMDA antagonist

1652Apamin

K+ channel blocker (small conductance, Ca2+-dependent)

12242-APB

IP3 receptor antagonist. Also TRP channel modulator

2511APC 366

Tryptase inhibitor

1208(2R,4R)-APDC

Highly selective group II agonist

2420[Pyr1]-Apelin-13

Potent peptide agonist for APJ receptor

3007Apelin-17 (human, bovine)

Endogenous APJ receptor agonist

2426Apelin-36 (human)

Endogenous APJ receptor agonist

2427Apelin-36 (rat, mouse)

Endogenous APJ receptor agonist

2151API-2

Selective inhibitor of Akt/PKB signaling. Antitumor and antiviral

1073(RS)-APICA

Selective group II antagonist

1227Apigenin

Protein kinase inhibitor

2073(R)-(-)-Apomorphine hydrochloride

Dopamine agonist; non-subtype-selective

2098Apoptosis Activator 2

Promotes apoptosome formation and activates caspase-9/caspase-3 pathway. Selectively induces tumor cell apoptosis

06663-AQC

5-HT3 antagonist

2292AQ-RA 741

Selective, high affinity M2 antagonist

2756Arachidonic acid (in TocrisolveTM 100)

Endogenous free fatty acid (in water-soluble emulsion)

3329N-Arachidonyl maleimide

Potent, competitive MAGL inhibitor

2836Arachidonyl serotonin

Dual FAAH inhibitor/TRPV1 antagonist

1814N-ArachidonylGABA

Inhibits pain in vivo

12982-Arachidonylglycerol

Endogenous cannabinoid agonist

1445N-Arachidonylglycine

Novel endocannabinoid. Suppresses pain in vivo

0928ARC 239 dihydrochloride

α2B antagonist

3321AR-C 66096 tetrasodium salt

Potent and selective P2Y12 antagonist

0389Arcaine sulfate

Competitive NMDA antagonist

1777Arctigenin

Potent MKK1 inhibitor. Also inhibits IκBα phosphorylation

2457Arcyriaflavin A

Potent cdk4/cyclin D1 and CaM Kinase II inhibitor. Antiviral agent (anti-HCMV)

0382Arecaidine but-2-ynyl ester tosylate

Muscarinic agonist

0383Arecaidine propargyl ester tosylate

Muscarinic agonist

0663L-Arginine

Endogenous substrate for NOS

1283ARL 67156 trisodium salt

Ecto-ATPase inhibitor

2699AR-M 1896

Selective GAL2 agonist

2621ARP 100

Selective inhibitor of MMP-2

2622ARP 101

Inhibitor of MMP-2

2668Artemisinin

Antimalarial; inhibits P-type ATPase (PfATP6) of P. falciparum

1354Arvanil

Potent CB1 and TRPV1 agonist. Also anandamide transport inhibitor

2446AS 101

Immunomodulator; inhibits IL-10 synthesis and potentiates IL-1α, IL-2 and TNF-α release

1968AS 19

Reported potent 5-HT7 agonist

3578AS 605240

Potent and selective PI 3-kinase γ (PI3Kγ) inhibitor

3737Asenapine maleate

Novel antipsychotic agent

0213D-Aspartic acid

NMDA agonist

0214L-Aspartic acid

NMDA agonist

3489Astemizole

Orally active, potent H1 antagonist. Also hERG K+ channel blocker.

1606Astressin

Potent CRF receptor antagonist

2391Astressin 2B

Selective CRF2 antagonist

0387(RS)-Atenolol

β1 antagonist

0393S-(-)-Atenolol

β1-antagonist. Active isomer of Cat.No. 0387

2937Atipamezole hydrochloride

Selective α antagonist

3776Atorvastatin hemicalcium salt

HMG-CoA reductase inhibitor

3245ATP disodium salt

P2 agonist

1107ATPA

Selective, potent GluR5 agonist

1912Atrial natriuretic factor (1-28) (rat)

Endogenous peptide regulating blood pressure

1906Atrial natriuretic factor (1-28) (human, porcine)

Endogenous peptide regulating blood pressure

1688Autocamtide-2-related inhibitory peptide

Selective CaM kinase II inhibitor

3126d[Cha4]-AVP

Potent and selective human V1B agonist

1639AY 9944 dihydrochloride

Inhibitor of hedgehog (Hh) signaling. Inhibits Δ7-dehydrocholesterol reductase

1487AY-NH2

Selective PAR4 agonist

2172AZ 10417808

Selective non-peptide caspase-3 inhibitor

3323AZ 10606120 dihydrochloride

Potent P2X7 receptor antagonist

3317AZ 11645373

Potent and selective human P2X7 antagonist

3771Azithromycin

Antibiotic; inhibits 50S ribosomal subunit formation and elongation at transpeptidation

Products by Catalog Number

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