| Cat. No. |
Product Name & Pharmacological Action |
| 2402 | MRS 2211 |
| Competitive P2Y13 antagonist |
| 2403 | MRS 3777 hemioxalate |
| High affinity, selective A3 antagonist |
| 2404 | Ambroxol hydrochloride |
| Na+ channel blocker |
| 2405 | p-DITC-APEC |
| Irreversible A2A agonist |
| 2408 | Ro 90-7501 |
| Inhibitor of Aβ42 fibril formation |
| 2409 | Conessine |
| Potent and selective H3 receptor antagonist |
| 2410 | L-371,257 |
| Potent and selective oxytocin receptor antagonist |
| 2411 | A-71623 |
| Potent and selective CCK1 agonist. Suppresses feeding |
| 2414 | H 1152 dihydrochloride |
| Selective rho-kinase (ROCK) inhibitor |
| 2415 | HA 1100 hydrochloride |
| Cell-permeable, selective Rho-kinase inhibitor |
| 2416 | BIBX 1382 dihydrochloride |
| Highly selective EGFR-kinase inhibitor |
| 2417 | BIBU 1361 dihydrochloride |
| Selective inhibitor of EGFR-kinase |
| 2418 | LY 303511 |
| Negative control of LY 294002 (Cat. No. 1130) |
| 2420 | [Pyr1]-Apelin-13 |
| Potent peptide agonist for APJ receptor |
| 2421 | Scriptaiδ |
| Histone deacetylase inhibitor |
| 2422 | AKTide-2T |
| Akt/PKB substrate (synthetic) |
| 2423 | DAPTA |
| Chemokine receptor 5 (CCR5) antagonist |
| 2424 | Amyloid β-peptide (1-40) (rat) |
| Amyloid β-protein fragment |
| 2425 | Amyloid β-peptide (1-42) (rat) |
| Predominant amyloid β-protein fragment |
| 2426 | Apelin-36 (human) |
| Endogenous APJ receptor ligand |
| 2427 | Apelin-36 (rat, mouse) |
| Endogenous APJ receptor ligand |
| 2429 | Fexofenadine hydrochloride |
| H1 receptor antagonist; non-sedating antiallergic agent |
| 2432 | Anagrelide hydrochloride |
| Potent PDE3 inhibitor |
| 2433 | L-759,633 |
| High affinity, selective CB2 agonist |
| 2434 | L-759,656 |
| Highly selective CB2 agonist |
| 2435 | CCT 018159 |
| Hsp90 inhibitor |
| 2436 | AC 55649 |
| Selective RARβ2 agonist |
| 2438 | TMPH hydrochloride |
| Neuronal nicotinic receptor antagonist |
| 2440 | NNC 26-9100 |
| Selective sst4 agonist |
| 2441 | JNJ 10191584 maleate |
| Selective H4 receptor antagonist; orally active |
| 2442 | CGP 53353 |
| Selective inhibitor of PKCβII |
| 2443 | RITA |
| p53-MDM2 interaction inhibitor; antitumour |
| 2444 | (1R,1'S,3'R/1R,1'R,3'S)-L-054,264 |
| Potent and selective sst2 agonist |
| 2445 | Obestatin (rat) |
| Endogenous anorexigenic peptide |
| 2446 | AS 101 |
| Immunomodulator; inhibits IL-10 synthesis and potentiates IL-1α, IL-2 and TNFα release |
| 2447 | Desmethyl-YM 298198 |
| Derivative of mGlu1 antagonist YM 298198 |
| 2448 | YM 298198 hydrochloride |
| Highly potent, selective non-competitive mGlu1 antagonist |
| 2450 | NF 157 |
| Selective P2Y11/P2X1 antagonist |
| 2451 | LY 344864 hydrochloride |
| Potent, selective 5-HT1F agonist |
| 2452 | LY 2183240 |
| Novel, potent anandamide uptake inhibitor. Inhibits FAAH |
| 2453 | LY 379268 |
| Highly selective group II mGlu agonist |
| 2456 | Co 101244 hydrochloride |
| Highly selective NR2B antagonist |
| 2457 | Arcyriaflavin A |
| Potent cdk4/cyclin D1 and CaM Kinase II inhibitor. Antiviral agent (anti-HCMV) |
| 2458 | ZM 447439 |
| Inhibits Aurora kinase B |
| 2459 | Tropisetron hydrochloride |
| Potent 5-HT3 receptor antagonist; orally active |
| 2460 | Lazabemide hydrochloride |
| Selective MAO-B inhibitor |
| 2463 | SCH 442416 |
| Very selective, high affinity A2A antagonist |
| 2464 | TNP-ATP triethylammonium salt |
| Potent, selective P2X antagonist |
| 2465 | SDZ WAG 994 |
| Potent, selective A1 agonist |
| 2466 | UK 14,304 tartrate |
| Water-soluble form of Cat. No. 0425 |
| 2467 | CGS 20625 |
| Selective central benzodiazepine receptor partial agonist |
| 2469 | IBC 293 |
| Selective agonist for the GPR109b (HM74) receptor. Antilipolytic |
| 2470 | Nimesulide |
| Cyclooxygenase-2 (COX-2) inhibitor |
| 2471 | ER 27319 maleate |
| Selective Syk kinase inhibitor |
| 2473 | GW 4064 |
| Selective farnesoid X receptor (FXR) agonist |
| 2474 | GW 3965 hydrochloride |
| Orally active liver X receptor (LXR) agonist |
| 2475 | ZM 323881 hydrochloride |
| Potent, selective inhibitor of VEGFR-2 |
| 2476 | SR 11302 |
| Inhibitor of AP-1 transcription factor; antitumour agent |
| 2477 | Proxyfan maleate |
| High affinity H3 ligand |
| 2478 | 2-Pyridylethylamine dihydrochloride |
| H1 receptor agonist |
| 2479 | JTE 907 |
| Selective CB2 receptor antagonist/inverse agonist |
| 2481 | JTC 801 |
| Selective ORL1 antagonist |
| 2483 | Costunolide |
| Inhibitor of human telomerase activity |
| 2484 | (±)-AC 7954 hydrochloride |
| Non-peptide UT receptor agonist |
| 2485 | Glycyl-H 1152 dihydrochloride |
| More selective analogue of Cat. No. 2414 |
| 2490 | (±)-Clopidogrel hydrochloride |
| Selective P2Y12 antagonist |
| 2491 | Xaliproden hydrochloride |
| Orally active, high affinity 5-HT1A agonist |
| 2492 | MNITMT |
| Immunosuppressant |
| 2493 | VUF 5681 dihydrobromide |
| Potent H3 receptor silent antagonist |
| 2494 | VUF 8430 dihydrobromide |
| Potent, high affinity H4 agonist |
| 2495 | Melperone hydrochloride |
| 5-HT2A/D2 receptor antagonist; neuroleptic |
| 2496 | DR 2313 |
| Potent PARP inhibitor |
| 2498 | PNU 120596 |
| Positive allosteric modulator of α7 nAChR; active in vivo |
| 2499 | ZM 306416 hydrochloride |
| Inhibitor of VEGF receptor tyrosine kinase |
| 2500 | Bay 59-3074 |
| CB1/CB2 receptor partial agonist |
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