Tocris Bioscience

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Product Pages Catalogue Numbers 1701 - 1800

Cat. No. Product Name & Pharmacological Action
1701A 77636 hydrochloride

Potent, selective D1-like agonist. Orally active
1702N6-Cyclopentyladenosine
Potent, selective A1 agonist
1704Ionomycin calcium salt
Calcium ionophore
17052-Chloro-N6-cyclopentyladenosine
Potent, selective A1 agonist
1706Acetaminophen
Cyclooxygenase inhibitor; may be selective for COX-3
1707Sulindac
Cyclooxygenase inhibitor (following metabolism to sulindac sulfide)
1708Indomethacin
Cyclooxygenase inhibitor (COX-1 > COX-2)
1709CL 218872
Benzodiazepine agonist
1710CV 1808
Adenosine A2 receptor agonist
1711TocriscreenTM Complete Collection
Compound library
1712TocriscreenTM Neuroscience Collection
Compound library
1713TocriscreenTM Signal Transduction Collection
Compound library
1714TocriscreenTM Adenosines
Collection of adenosine receptor and related compounds
1715TocriscreenTM Adrenergics
Collection of adrenoceptor and related compounds
1716TocriscreenTM Cannabinoids
Collection of cannabinoid receptor and related compounds
1717TocriscreenTM Cholinergics
Collection of cholinergic receptor and related compounds
1718TocriscreenTM Dopaminergics
Collection of dopamine receptor and related compounds
1719TocriscreenTM Enzyme Inhibitors
Collection of enzyme inhibitors
1720TocriscreenTM GABA/Glycine Ligands
Collection of GABA/glycine receptor and related compounds
1721TocriscreenTM Glutamate Ligands
Collection of glutamate receptor and related compounds
1722TocriscreenTM Histaminergics
Collection of histamine receptor and related compounds
1723TocriscreenTM Imidazolines
Collection of imidazoline receptor and related compounds
1724TocriscreenTM Ion Channel Modulators
Collection of ion channel modulators
1725TocriscreenTM Melatonergics
Collection of melatonin receptor and related compounds
1726TocriscreenTM Nitric Oxide
Collection of nitric oxide tools
1727TocriscreenTM Opioids
Collection of opioid receptor and related compounds
1728TocriscreenTM Peptide Receptor Ligands
Collection of peptide receptor and related compounds
1729TocriscreenTM Prostanoids
Collection of prostanoid receptor and related tools
1730TocriscreenTM Purinergics
Collection of purinergic receptor and related compounds
1731TocriscreenTM Retinoids and PPARs
Collection of retinoid and PPAR receptor and related tools
1732TocriscreenTM Serotonergics
Collection of 5-HT receptor and related compounds
1733TocriscreenTM Sigma Ligands
Collection of sigma receptor and related compounds
1734TocriscreenTM Calcium Signalling
Collection of calcium signalling tools
1735TocriscreenTM Cyclic Nucleotide Tools
Collection of cyclic nucleotide tools
1736TocriscreenTM Lipid Signalling
Collection of lipid signalling tools
1737TocriscreenTM Protein Kinase/Phosphatase Tools
Collection of protein kinase/protein phosphatase tools
1738TocriscreenTM Cell Cycle and Apoptosis
Collection of cell cycle and apoptosis tools
1739TocriscreenTM Steroid Hormones
Collection of steroid hormone receptor and related tools
1740TocriscreenTM Vanilloids
Collection of vanilloid receptor and related tools
1741TocriscreenTM Miscellaneous Signalling
Collection of miscellaneous signalling tools
1742R-96544 hydrochloride
Potent, selective 5-HT2A antagonist
1743Bay 11-7085
Irreversible inhibitor of TNF-α-induced IκBα phosphorylation
1744Bay 11-7821
Irreversible inhibitor of TNF-α-induced IκBα phosphorylation
1746Nemonapride

Highly potent D2-like antagonist. Also 5-HT1A agonist
1747Isoproterenol hydrochloride

Standard selective β-adrenoceptor agonist
1748MG 132
Proteasome and calpain inhibitor. Inhibits NF-κB activation
1749HexylHIBO
Group I mGlu antagonist
1750(S)-HexylHIBO
Group I mGlu antagonist
1757ALX 5407 hydrochloride
Selective non-transportable GlyT1 inhibitor
1758PETCM
Activator of caspase-3
1759Nilutamide
Androgen receptor antagonist. Orally active
1760(±)-Blebbistatin
Selective inhibitor of myosin II
1761Baicalein
5- and 12-Lipoxygenase inhibitor
1762Acifran
Hypolipidaemic agent; agonist for the GPR109a (HM74A) and GPR109b receptors
1763BAM (8-22)
Selective agonist for the sensory neuron specific receptor (SNSR)
1764Hemopressin
Bioactive substrate for endopeptidase 24.15, neurolysin and ACE
1765UBP 282
AMPA/kainate antagonist; distinguishes between motoneuron and dorsal root kainate receptors
1766UBP 301
Kainate receptor antagonist
1767Zimelidine dihydrochloride
Selective 5-HT uptake inhibitor
1768Fumagillin
Methionine aminopeptidase-2 inhibitor
1769Flurbiprofen
Cyclooxygenase inhibitor
1770Deguelin
Anticancer and antiviral agent; chemopreventive and proapoptotic
1771S 14506 hydrochloride
Highly potent 5-HT1A agonist; displays unique binding mechanism
1772Urapidil hydrochloride
α1 antagonist. Also 5-HT1A receptor agonist
1774Dynamin inhibitory peptide
Dynamin inhibitor
1775Dynamin inhibitory peptide, myristoylated
Cell-permeable dynamin inhibitor
1776Dynamin inhibitory peptide, myristoylated (control)
Control peptide version of Cat. Nos. 1774 and 1775
1777Arctigenin
Inhibitor of IκBα phosphorylation. Also inhibits MKK1
1778Ro 106-9920
Inhibitor of NF-κB activation
1779NNC 711
Selective inhibitor of GAT-1
1780NNC 63-0532
Potent non-peptide ORL1 agonist; brain penetrant
1781ACPA (in TocrisolveTM 100)

Potent, selective CB1 agonist (in water-soluble emulsion)
1782(R)-(+)-Methanandamide (in TocrisolveTM 100)

Potent and selective CB1 agonist (in water-soluble emulsion)
1783JWH 133 (in TocrisolveTM 100)

Potent, selective CB2 agonist (in water-soluble emulsion)
1784Spantide I
Selective NK1 antagonist
1785Bax inhibitor peptide V5
Inhibitor of Bax-mediated apoptosis
1786Bax inhibitor peptide P5
Inhibitor of Bax-mediated apoptosis
1787Bax inhibitor peptide, negative control
Negative control peptide for Cat. Nos. 1785 and 1786
1788GRP (porcine)
Endogenous GRP receptor agonist
1789GRP (human)
Endogenous GRP receptor agonist
1790Pseudo RACK1
Protein kinase C activator peptide (attached to cell permeable vector)
1791PKC z pseudosubstrate
PKC z inhibitor peptide (attached to cell-permeable vector)
1792PKC β pseudosubstrate
Selective cell-permeable PKC inhibitor peptide (attached to vector)
1793AF 12198
Potent, selective human type I IL-1 receptor antagonist
1794Ro 26-4550 trifluoroacetate
Competitive inhibitor of IL-2/ IL-2Rα receptor interaction
1795Zacopride hydrochloride
Highly potent 5-HT3 receptor antagonist. Also 5-HT4 agonist
1797OMDM-2

Potent inhibitor of anandamide uptake
1798Gabexate mesylate
Serine proteinase inhibitor; inhibits thrombin, trypsin, kallikrein and plasmin
1799WKYMVM
Selective FPRL1 and FPRL2 receptor agonist
1800WKYMVm
FPR, FPRL1 and FPRL2 receptor agonist
 
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