Tocris Bioscience

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Product Pages Catalogue Numbers 1601 - 1700

Cat. No. Product Name & Pharmacological Action
1601Pep1-TGL
GluR1 subunit C-terminus peptide analogue
1602Pep1-AGL
Analogue of Cat. No. 1601
1603NKH 477
Water-soluble adenylyl cyclase activator
1604Urocortin (human)
Endogenous CRF agonist
1605Urocortin (rat)
Endogenous CRF agonist
1606Astressin
Potent CRF receptor antagonist
1607CRF (6-33)
CRF-binding protein inhibitor
1608Stressin I
CRF1 agonist
1609Sauvagine
CRF agonist
1610Rottlerin
Reported PKCδ inhibitor
1611Lamotrigine
Inhibits glutamate release. Anticonvulsant
1612SB 269970 hydrochloride
Potent selective 5-HT7 antagonist. Brain penetrant
1614SB 431542
Potent, selective inhibitor of TGF-β receptor ALK5, and ALK4 and 7
1615SB 366791
Potent, selective, competitive TRPV1 (VR1) antagonist
1616SB 216763
Potent selective GSK-3 inhibitor
1617SB 415286
Potent selective GSK-3 inhibitor
1618Peptide YY (3-36)
Selective Y2 receptor agonist
1619[Orn8]-Urotensin II
Urotensin II (UT) receptor partial agonist
1620Alprostadil
Prostaglandin. Vasodilator and anti-platelet agent in vivo
1621Streptozocin
DNA alkylator; antitumour and induces diabetes
1622Remacemide hydrochloride
NMDA antagonist; blocks ion channel and allosteric modulatory site
1623Cyclopamine
Inhibitor of hedgehog (hh) signalling
16242-Methylthio-ADP trisodium salt
Potent agonist for P2Y1, P2Y12 and P2Y13
1625DFB
Allosteric potentiator at mGlu5
1626Calphostin C
Potent, selective and photo-dependent PKC inhibitor
1628NPC 15437 dihydrochloride
Selective protein kinase C inhibitor
1632MEN 10376
Potent, selective NK2 antagonist
1633MEN 10627
Potent, selective NK2 antagonist
1634Y-29794 oxalate
Prolyl endopeptidase inhibitor
1635RP 67580
Potent and selective NK1 antagonist
1636IEM 1460
Open-channel blocker of AMPA currents; selective for non-GluR2-containing receptors
1638U 18666A
Inhibitor of hedgehog (hh) signalling. Also inhibits cholesterol synthesis
1639AY 9944 dihydrochloride
Inhibitor of hedgehog (hh) signalling.  Inhibits D7-dehydrocholesterol reductase
1640[bAla8]-Neurokinin A(4-10)
NK2 agonist
1641OLDA
Potent, selective endogenous TRPV1 (VR1) agonist
1642Urotensin II (human)
Endogenous vasoactive agonist for the UT-II receptor
1643D-64131
Inhibitor of tubulin polymerisation. Antitumour in vivo
16458CPT-2Me-cAMP, sodium salt
Selective Epac activator
1646Lonidamine
Mitochondrial hexokinase inhibitor
1650BAM 22P
Opioid receptor agonist. Also agonist at the sensory neuron specific receptor (SNSR)
1652Apamin
K+ channel blocker (small conductance, Ca2+-dependent)
1655O-2050

CB1 silent antagonist

1657Ginkgolide B
PAF receptor antagonist
1658GR 125487 sulfamate
Potent, selective 5-HT4 antagonist. Active in vivo
1659Fenoldopam hydrochloride

Selective D1-like partial agonist

1660Salmeterol

Potent β2 agonist; long acting

1661SB 206553 hydrochloride
Potent, selective 5-HT2C/5-HT2B antagonist. Orally active
1662SKF 77434 hydrobromide

Selective D1-like partial agonist

1663BW 373U86
Potent, selective non-peptide δ-opioid agonist
1664GW 1929
Selective PPARγ agonist. Orally active
1667GR 94800
Potent, selective NK2 antagonist
1668GR 64349
Potent, selective NK2 agonist
1669GR 73632
Potent, selective NK1 agonist
1670GR 82334
Tachykinin NK1 receptor antagonist
1671PD 102807

Selective M4 antagonist

1672RU 28318, potassium salt
Potent, selective mineralocorticoid receptor antagonist
1673Cl-HIBO
Subtype-selective AMPA agonist (GluR1 and GluR2)
1674LE 300

Potent and selective dopamine D1 antagonist

1675YM 90709
Interleukin-5 receptor antagonist
1676T 0156 hydrochloride
Highly potent, selective PDE5 inhibitor
1677GW 7647
Highly selective, potent PPARα agonist. Orally active
1682PIT
P2Y ligand; displays mixed antagonism/potentiation
1683K 252a
Protein kinase inhibitor
1684TocrisolveTM 100

Water-soluble emulsion; negative control for Cat. Nos. 1017, 1685, 1686, 1781, 1782 and 1783

1685AM 404 (in TocrisolveTM 100)

Anandamide transport inhibitor (in water-soluble emulsion)

1686VDM 11 (in TocrisolveTM 100)

Potent, selective anandamide transport inhibitor (in water-soluble emulsion)

1688Autocamtide-2-related inhibitory peptide
Selective CaM kinase II inhibitor
1690SCH 28080
H+,K+-ATPase inhibitor
1691NECA
Adenosine receptor agonist
1692Cilostazol
PDE3A inhibitor. Also adenosine uptake inhibitor
1694Ibudilast
PDE inhibitor (non-selective)
1695Cisapride
5-HT4 agonist; stimulates intestinal ACh release
1697Noscapine hydrochloride
Tubulin inhibitor; induces apoptosis
1698L-655,240
Potent, selective thromboxane A2/prostaglandin endoperoxide antagonist
1699CGS 15943
Potent adenosine receptor antagonist
1700BIIE 0246 formate
Potent, selective non-peptide NPY Y2 antagonist
 
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