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Product Pages Catalogue Numbers 1301 - 1400

Cat. No. Product Name & Pharmacological Action
1302(S)-3,4-DCPG
Potent, selective mGlu8a agonist
1304BW-B 70C
5-Lipoxygenase inhibitor
1305Monastrol
Selective inhibitor of mitotic kinesin Eg5
1307Ciglitazone
Selective PPARγ agonist
1308[Nphe1]Nociceptin(1-13)NH2
Selective, competitive nociceptin antagonist
1309PPNDS
Potent, selective P2X1 antagonist
1310UCL 1684
Highly potent blocker of SKCa
1311MK 886
Inhibitor of 5-lipoxygenase-activating protein (FLAP)
1312WY 14643
Selective PPARα agonist
1316Tertiapin-Q
Potent, selective inhibitor of inward-rectifier K+ channels
1317CP 94253 hydrochloride
Potent, selective 5-HT1B agonist
1318ACPA

Potent, selective CB1 agonist

1319ACEA

Potent, highly selective CB1 agonist

1321ZM 336372
Potent, selective c-Raf inhibitor
1322GR 113808
Potent, selective 5-HT4 antagonist
1323Butabindide oxalate
CCK-inactivating serine peptidase inhibitor
1324RX 821002 hydrochloride

Potent, selective α2D antagonist

1325RS 100329 hydrochloride
Potent, subtype selective α1A antagonist
1326BADGE
PPARγ antagonist
1327L-655,708
Selective for α5-containing GABAA receptors
1328Flumazenil
Benzodiazepine antagonist
1329Ryanodine
Ca2+ release inhibitor
1330Chelerythrine chloride
Potent protein kinase C inhibitor
1331Lavendustin A
EGFR, p60c-src inhibitor
1333cAMPS-Sp, triethylammonium salt
Cell-permeable cAMP analogue
1334Bafilomycin A1
H+-ATPase (vacuolar) inhibitor
1336Calyculin A
Protein phosphatase 1 and 2A inhibitor
1337cAMPS-Rp, triethylammonium salt
cAMP antagonist
1339Anandamide

Endogenous CB receptor agonist

1341JWH 015

Selective CB2 agonist

1343JWH 133

Potent, selective CB2 agonist

1344SAMS Peptide
AMP-activated protein kinase substrate
1345AF-DX 384

Potent M2/M4 antagonist

1346des-Gln14-Ghrelin (rat)
Endogenous ligand for GHS receptor
1347Nafadotride

Highly potent, preferential D3 antagonist

1348UB 165 fumarate

Subunit selective nAChR agonist

1349(R)-(-)-Rolipram
More active enantiomer of Cat. No. 0905
1350(S)-(+)-Rolipram
Less active enantiomer of Cat. No. 0905
1352Phospho-Glycogen Synthase Peptide-2 (substrate)
Glycogen synthase kinase-3 substrate (synthetic)
1353Akt/SKG Substrate Peptide
Akt/PKB substrate (synthetic)
1354Arvanil
Potent CB1 and TRPV1 (VR1) agonist/anandamide transport inhibitor
1355P1075
Potent KATP channel opener
1356MG 624

α7 neuronal nicotinic receptor antagonist

1357U 99194 maleate

Potent, selective D3 antagonist

1358Nociceptin (1-13)NH2
Potent ORL1 agonist
1359VUF 5574
Potent, selective hA3 antagonist
1361PD 123319 ditrifluoroacetate
Potent, selective non-peptide AT2 antagonist
13625'-Iodoresiniferatoxin
Potent, silent TRPV1 (VR1) antagonist
1363PD 81723
Allosteric potentiator of A1 receptors
1364Colchicine
Inhibitor of tubulin
1365[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] -hPancreatic Polypeptide
Potent, selective neuropeptide Y Y5 agonist
1366ZM 449829
Potent, selective Jak3 inhibitor
1367ZM 39923 hydrochloride
Potent, selective Jak3 inhibitor
1368Geldanamycin
Selective Hsp90 inhibitor
1369UBP1112
Group III mGlu antagonist
1370Sphingosine-1-phosphate
Bioactive lipid, binds EDG receptors
1371SB 200646 hydrochloride
5-HT2C/2B antagonist
1372SB 204741
Potent, selective 5-HT2B antagonist
1375SB 228357
5-HT2C/2B antagonist/inverse agonist
1376SB 218795
Potent, selective non-peptide NK3 antagonist
1377Cromakalim
KATP channel opener
1378Levcromakalim
KATP channel opener. Active enantiomer of Cat. No. 1377
1379SB 221284
Potent, selective 5-HT2C/2B antagonist
1380PMPA (NAALADase inhibitor)
Highly potent, selective NAALADase (GCP II) inhibitor
1381GW 5074
Potent, selective cRaf1 kinase inhibitor
1382L-152,804
Potent, selective non-peptide NPY Y5 antagonist
1383BML-190

Potent, selective CB2 ligand

1384McN-A 343
Selective M1 muscarinic agonist
1385MRS 1334
Potent, highly selective hA3 antagonist
1386[Ala11,22,28]VIP
Potent, highly selective VPAC1 agonist
1387Ac-RYYRWK-NH2
Potent, selective ORL1 partial agonist peptide
1390(-)-Cytisine

Potent, selective neuronal nicotinic agonist

1391NF 449
Highly selective P2X1 antagonist
1392VDM 11

Potent, selective anandamide transport inhibitor

1393SB 222200
Potent, selective non-peptide NK3 antagonist. Brain penetrant
1394(RS)-3,4-DCPG
AMPA/NMDA antagonist/mGlu8 agonist. Anticonvulsant
1395(R)-3,4-DCPG
AMPA antagonist/weak NMDA antagonist
1396Fenretinide
Synthetic retinoid. Potent anti-cancer agent
1397PP 1
Potent, selective Src inhibitor
1398Kenpaullone
Potent cyclin-dependent kinase inhibitor. Also inhibits GSK-3
1399CP 339818 hydrochloride
Non-peptide, potent Kv1.3 channel blocker
1400SCH 202676 hydrobromide
Inhibitor of ligand binding to G-protein-coupled receptors
 
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