Tocris Bioscience

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Product Pages Catalogue Numbers 1001 - 1100

Cat. No. Product Name & Pharmacological Action
1001Chlorisondamine diiodide

Nicotinic antagonist; slow offset

1002L-745,870 trihydrochloride

Highly selective D4 antagonist

1003L-741,626

High affinity D2 antagonist

1004L-741,742 hydrochloride

Highly selective D4 antagonist

1006BMY 7378 dihydrochloride
Selective α1D antagonist, 5-HT1A partial agonist
1007N-Desmethylclozapine
5-HT2C antagonist
1008SNC 121
Potent analogue of Cat. No. 0764
1009E4CPG
Group I/group II mGlu antagonist
1014QX 314 bromide
Na+ channel blocker
1015RS 16566 dihydrochloride
5-HT3 ligand. Also shows affinity for zacopride binding site
1017Anandamide (in TocrisolveTM 100)

Endogenous CB receptor agonist (in water-soluble emulsion)

1018LY 225910
Potent CCK2 antagonist
1019LY 235959
Competitive NMDA antagonist
1024CGP 20712 dihydrochloride

Highly potent and selective β1 antagonist

1025Nisoxetine hydrochloride

Noradrenaline re-uptake inhibitor

1026HomoAMPA
Potent, highly selective mGlu6 agonist
1027PHCCC
Potent group I mGlu antagonist
1028CPCCOEt
Selective non-competitive mGlu1 receptor antagonist
1029Methyllycaconitine citrate

α7 neuronal nicotinic receptor antagonist

1030Guanfacine hydrochloride

α2A agonist

1031Piribedil hydrochloride

Dopamine agonist

1032CP 93129 dihydrochloride
5-HT1B agonist
1033Fluvoxamine maleate
5-HT re-uptake inhibitor
10344-P-PDOT
MT2 antagonist
10358-M-PDOT
Melatonin agonist
1036ZM 241385
Potent, highly selective A2A antagonist
1037PD 153035 hydrochloride
EGFR-kinase inhibitor
1038WIN 55,212-2 mesylate

Highly potent cannabinoid agonist

1040TPMPA
Selective GABAC antagonist
10411-EBIO
Activator of epithelial Kca channels
1042N-Methyllidocaine iodide
Enhances biosynthesis of phosphatidylinositol
1043QX 222
Na+ channel blocker
1044NBQX disodium salt
More water soluble form of (0373)
1045CNQX disodium salt
More water soluble form of (0190)
1046Zardaverine
PDE3/4 inhibitor
1047ICI 182,780
Estrogen receptor antagonist
10481-BCP
Modulates AMPA-mediated responses
1049CHPG
mGlu5 selective agonist
1050RS 102221 hydrochloride
Selective 5-HT2C antagonist
1051Zinterol hydrochloride
Selective β2 agonist
1052A 61603 hydrobromide
α1A agonist
1053RJR 2403 fumarate

CNS selective nicotinic agonist

1054GR 55562 dihydrochloride
5-HT1B antagonist
1055Endomorphin-1
Potent and selective μ agonist
1056Endomorphin-2
Potent and selective μ agonist
1057WIN 64338 hydrochloride
Bradykinin B2 antagonist
1058L-3'-F2CCG-I
Potent group I/group II agonist
1059BW 723C86 hydrochloride
5-HT2B agonist
1060(S)-(-)-Pindolol

More active enantiomer

1061(-)-Quinpirole hydrochloride

Selective D2-like agonist

10622-Methylthioadenosine triphosphate tetrasodium salt
P2 purinergic agonist
1063CGS 21680 hydrochloride
A2A agonist
1064Methysergide maleate
5-HT1/5-HT2 antagonist
1065PD 168077 maleate

High affinity, selective D4 agonist

1066IB-MECA
A3 selective agonist
1067Oxotremorine M

Muscarinic agonist

1068Senktide
Tachykinin NK3 agonist
1069Tetrodotoxin citrate
Citrate salt of Cat. No. 1078
1070Zolantidine dimaleate
Potent, centrally active H2 antagonist
1071Pirenzepine dihydrochloride

Selective M1 muscarinic antagonist

1072AGN 192403 hydrochloride
I1 selective ligand
1073(RS)-APICA
Selective group II antagonist
1074(RS)-AMPA hydrobromide
More water soluble form of Cat. No. 0169
1075Nifedipine
Ca2+ channel blocker (L-type)
1076Ouabain
Na+,K+-ATPase inhibitor
1077(-)-Lobeline hydrochloride

Nicotinic agonist

1078Tetrodotoxin
Na+ channel blocker
1079(+)-SK&F 10047 hydrochloride
σ1 selective agonist
1080(R)-(+)-8-Hydroxy-DPAT hydrobromide
More active enantiomer
1081SKF 89976A hydrochloride
Potent GABA uptake inhibitor. Penetrates blood brain barrier
1082CFM-2
Non-competitive AMPA antagonist
1084ω-Conotoxin MVIIC
Ca2+ channel blocker (N, P and Q-type)
1085ω-Conotoxin GVIA
Ca2+ channel blocker (N-type)
1086Iberiotoxin
K+ channel blocker (high conductance, Ca2+-dependent)
1087Charybdotoxin
K+ channel blocker (high conductance, Ca2+-dependent)
1088CGP 54626 hydrochloride
Potent, selective GABAB antagonist
10898-Bromo-cGMP, sodium salt
cGMP analogue
1091BU 226 hydrochloride
Potent, highly selective I2 ligand
1092[Phe1Y(CH2-NH)Gly2]Nociceptin(1-13)NH2
Selective nociceptin agonist
1093Pirfenidone
Antifibrotic agent; regulates cytokine levels in vivo
1094Zopiclone
Benzodiazepine agonist
1095(R)-(-)-Deprenyl hydrochloride
MAO-B inhibitor
1097Taxol
Promotes assembly and inhibits disassembly of microtubules
1098Tranilast
Anti-allergic, inhibits release from mast cells
1099Forskolin
Adenylyl cyclase activator
1100Camptothecin
DNA topoisomerase inhibitor
 
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