Tocris Bioscience

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Product Pages Catalogue Numbers 0801 - 0900

Cat. No. Product Name & Pharmacological Action
0803MSOP
Specific group III mGlu antagonist
0805(S)-3,5-DHPG
Active enantiomer of (0342)
0806Gabapentin
Anticonvulsant. Increases brain GABA
0807THIP hydrochloride
GABAA agonist
0808Vigabatrin
GABA-T inhibitor
0811(±)-threo-3-Methylglutamic acid
EAAT2 and EAAT4 blocker
0817(2R,3S)-Chlorpheg
Weak NMDA antagonist
0820ICI 174,864
δ selective peptide antagonist
0821ICI 118,551 hydrochloride

Very selective β2 antagonist

0822ICI 204,448 hydrochloride
κ agonist, acts peripherally
0823ICI 216,140
Potent Bombesin/Gastrin releasing peptide antagonist
0824Clofibrate
PPAR agonist
0825Clofibric acid
PPAR agonist
0826Tiotidine
Potent, selective H2 antagonist
0827ICI 154,129
δ selective peptide antagonist
0829Pronethalol hydrochloride

β antagonist

0830Primidone
Potentiates GABAA receptor function
0831Practolol

β1 antagonist

0832ICI 89406

β antagonist

0833ICI 162,846
Potent H2 antagonist, active in vivo
0834(S)-(-)-Propranolol hydrochloride

More active enantiomer

0835(R)-(+)-Propranolol hydrochloride

Less active enantiomer

0836ICI 185,282
Potent thromboxane receptor antagonist
0837ICI 192,605
Potent thromboxane A2/TP receptor antagonist
0839DHBP dibromide
Ca2+ release inhibitor
0840Loperamide hydrochloride
Peripherally acting μ agonist. Also Ca2+ channel blocker
0841DTG
High affinity ligand (σ1 = σ2)
0842Agmatine sulfate

α2 ligand. Also imidazoline ligand

0843Oxotremorine sesquifumarate

Muscarinic agonist

0845Evans Blue tetrasodium salt
Potent inhibitor of L-glutamate uptake into synaptic vesicles
0846Chicago Sky Blue 6B
Potent inhibitor of L-glutamate uptake into synaptic vesicles
0847Statil
Aldose reductase inhibitor
0851Propranolol glycol

Propranolol metabolite

0853MPPG
Group III/group II mGlu antagonist. More selective for group III than group II
0854MSPG
Group II/group III mGlu antagonist
0855MTPG
Group II/group III mGlu antagonist. More selective for group II than group III
0860tADA
Group I agonist; some mGlu5 selectivity
0864GR 46611
5-HT1D agonist
0867Aniracetam
Desensitization inhibitor (AMPA > kainate)
0868L-732,138
Potent, selective NK1 antagonist
0869Felbamate
NMDA antagonist, acts glycine site
0870MDL 11,939
5-HT2 antagonist
0871AMT hydrochloride
Potent, selective iNOS inhibitor
0872Cypermethrin
Calcineurin inhibitor (protein phosphatase 2B)
0873EIT hydrobromide
Selective iNOS inhibitor, acts arginine binding site
0875μ-CPP hydrochloride
5-HT2B/2C receptor agonist
0876AM 92016 hydrochloride
K+ channel blocker (KV)
0877Luzindole
Competitive melatonin MT1/MT2 antagonist
0878Oleamide
Potentiator at 5-HT2A/2C receptors. Also CB1 agonist
0879Palmitoylethanolamide
Agonist for putative CB2-like receptor. FAAH and PAA substrate
0880ODQ
Selective inhibitor of NO-sensitive guanylyl cyclase
0881Chlormethiazole hydrochloride
Potentiates GABAA receptor function
0882ZM 226600
KATP channel opener
0883BD 1063 dihydrochloride
Selective σ1 ligand, putative antagonist
0884Dihydrexidine hydrochloride

Selective D1-like agonist

0885Guanabenz acetate

α2 agonist. Also I2 selective ligand

0888Cirazoline hydrochloride
Selective α1 agonist
0889RS 45041-190 hydrochloride
High affinity I2 ligand. Highly selective
0890Amiloride hydrochloride
Na+ channel blocker. Also I2 imidazoline ligand
0891Rauwolscine hydrochloride

α2 antagonist

0892Naltriben mesylate
Standard δ2 selective antagonist
0894(RS)-(±)-Sulpiride

Standard selective D2-like antagonist

0895(S)-(-)-Sulpiride

Standard selective D2-like antagonist

0896GR 135531
High affinity melatonin MT3 ligand
0897S-Isopropylisothiourea hydrobromide
iNOS inhibitor, acts arginine binding site
0899BNTX maleate
Standard δ1 selective antagonist
0900MRS 2179 tetrasodium salt
Selective P2Y1 antagonist
 
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