Tocris Bioscience

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Product Pages Catalogue Numbers 0601 - 0700

Cat. No. Product Name & Pharmacological Action
0601Nitrendipine
Ca2+ channel blocker (L-type)
06027-Nitroindazole
Non-selective NOS inhibitor
0603SNOG
NO carrier. Breaks down to release NO
0604Nicergoline

α antagonist

0605(±)-Octanoylcarnitine chloride
Intermediate in lipid metabolism
0606OBAA
Phospholipase A2 inhibitor
060717-ODYA
LTB-ω-Hydroxylase inhibitor
0609(±)-Palmitoylcarnitine chloride
Protein kinase C inhibitor
0610Parthenolide
5-HT release inhibitor
0611(±)-Propionylcarnitine chloride
Intermediate in lipid metabolism
0616AG 556
EGFR-kinase inhibitor
0618AG 555
Potent EGFR-kinase inhibitor
0619AG 494
Potent EGFR-kinase inhibitor
06204-PPBP maleate
Specific σ ligand, NMDA antagonist
0622Physostigmine hemisulfate

Cholinesterase inhibitor

0623Prazosin hydrochloride
α1 antagonist. MT3 antagonist
0624Propranolol hydrochloride

β antagonist

0625PPADS tetrasodium salt
P2 purinergic antagonist
06272-[(4-Phenylpiperazin-1-yl)methyl]-2,3-dihydroimidazo[1,2-c]quinazolin-5(6H)-one
Potent, selective α1 antagonist
0629Quipazine dimaleate
5-HT3 agonist
0630Rosmarinic acid
Anti-inflammatory, cytostatic and anti-viral
0631Spiroxatrine

Potent α2 ligand

0633D-erythro-Sphingosine (synthetic)
Protein kinase C inhibitor
0634Salbutamol hemisulfate

β agonist (β2>β1)

0635Synthalin sulfate
Non-competitive NMDA antagonist
0636Salsolinol-1-carboxylic acid
Endogenous amino acid
0638CGS 12066B dimaleate
5-HT1B agonist
0640MDL 72222
5-HT3 antagonist
0641Tropanyl-3,5-dimethylbenzoate
5-HT3 antagonist
0644Thioperamide maleate
H3/H4 antagonist, active in vivo
06452-(1-Thienyl)ethyl 3,4-dihydroxybenzylidenecyanoacetate
5-, 12-, 15-Lipoxygenase inhibitor
0646HTMT dimaleate
H1 / H2 agonist
0649(S)-Timolol maleate

β1 antagonist

0650Trimethoprim
Dihydrofolate reductase inhibitor
0652Thalidomide
TNF-α synthesis inhibitor
0653(±)-Vesamicol hydrochloride

Inhibits ACh transport

0654Verapamil hydrochloride
Ca2+ channel blocker (L-type)
0655Zolpidem
Benzodiazepine agonist
0658FGIN-1-27
Potent, specific ligand for mitochondrial DBI receptor
0659FGIN-1-43
Potent, specific ligand for mitochondrial DBI receptor
0660Mepyramine maleate
Selective H1 inverse agonist
06612-[[4-(2-Methoxyphenyl)piperazin-1-yl] methyl]-6-methyl-2,3-dihydroimidazo[1,2c]quinazolin-5(6H)-one
Potent, selective α1 antagonist and σ2 ligand
0662trans-Triprolidine hydrochloride
Standard H1 antagonist, highly potent
0663L-Arginine
Endogenous substrate for NOS
0664L-NNA
NOS inhibitor (nNOS = eNOS >> iNOS)
0665L-NAME hydrochloride
Non-selective NOS inhibitor
06663-(4-Allylpiperazin-1-yl)-2-quinoxalinecarbonitrile maleate
5-HT3 antagonist
0668Amthamine dihydrobromide
Highly selective standard H2 agonist
0670PK 11195
Antagonist at peripheral BDZ receptors
0671AH 6809
EP1 and EP2 receptor antagonist
0673L-Canavanine sulfate
iNOS inhibitor
0674Dequalinium dichloride
K+ channel blocker (SKCa)
0675NPC 15199
Novel anti-inflammatory agent
0677Naltrexone hydrochloride
Broad spectrum opioid antagonist
0678(+)-AJ 76 hydrochloride

Antagonist; preferential action at D2-like autoreceptors

06802-Phenylmelatonin
Potent melatonin agonist
0681L-690,330
Inositol monophosphatase inhibitor
0682L-690,488
Cell permeable prodrug of the IMPase inhibitor L-690,330 (Cat. No. 0681)
0683iso-PPADS tetrasodium salt
P2X purinergic antagonist
0684(±)-Epibatidine

Very potent nicotinic agonist

0685Diltiazem hydrochloride
Ca2+ channel blocker (L-type)
0686Galanthamine hydrobromide

Cholinesterase inhibitor

0687Danazol

Anterior pituitary suppressant

0690Clonidine hydrochloride
α2 agonist. Also I1 ligand
0691Dipyridamole
Adenosine transport inhibitor
0692Ipratropium bromide

Muscarinic antagonist

0693Pancuronium dibromide

Nicotinic (neuromuscular) antagonist

0694Pilocarpine hydrochloride

Muscarinic agonist

0695Retinoic acid
Endogenous retinoic acid receptor agonist. Also modulates PPARδ
0699BRL 52537 hydrochloride
Potent and selective κ agonist
 
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