Tocris Bioscience

Site Map

Product Pages Catalogue Numbers 0401 - 0500

Cat. No. Product Name & Pharmacological Action
0405β-CCB
Benzodiazepine inverse agonist, putative endogenous ligand
0411MDL 73005EF hydrochloride
Potent and selective 5-HT1A partial agonist
0412MDL 72832 hydrochloride
Potent 5-HT1A ligand
0414AG 490
EGFR-kinase inhibitor. Also Jak2, Jak3 inhibitor
0415Ro 20-1724
PDE4 inhibitor
0416YS-035 hydrochloride
Inhibits K+ outward/pacemaker current
0417(RS)-Baclofen
Selective GABAB agonist
0420GBR 13069 dihydrochloride

Potent dopamine uptake inhibitor

0421GBR 12909 dihydrochloride

Selective DA uptake inhibitor. Also σ ligand

0424Benzoquinonium dibromide

Nicotinic antagonist

0425UK 14,304

α2 agonist

0426L-693,403 maleate
High affinity σ ligand
0427Bromocriptine mesylate

Selective D2-like agonist

0430SC-10
Protein kinase C activator
0431ML 9 hydrochloride
Myosin light chain kinase inhibitor
0432MY-5445
PDE5 inhibitor
0433SC-9
Protein kinase C activator
0435Cimaterol

β agonist

0438Etazolate hydrochloride
PDE4 inhibitor
0439DPCPX
A1 selective antagonist
0440m-Chlorophenylbiguanide hydrochloride
Potent and specific 5-HT3 agonist
04424-Chlorophenylguanidine hydrochloride
Urokinase inhibitor
04436-Chloromelatonin
Melatonin agonist
0444Clozapine
Dopamine antagonist with some D4 selectivity. Also muscarinic antagonist and 5-HT ligand
0448Calpeptin
Calpain and cathepsin L inhibitor
0452CCCP
Oxidative phosphorylation uncoupler
0453FCCP
Oxidative phosphorylation uncoupler
0454Carbetapentane citrate
High affinity σ1 ligand
0455(S)-(-)-Carbidopa
Aromatic L-amino acid decarboxylase inhibitor
0456Chlormezanone
Skeletal muscle relaxant
0457Clomipramine hydrochloride
5-HT re-uptake inhibitor
04585-Carboxamidotryptamine maleate
5-HT1 agonist. Also has high affinity for 5-ht5A and 5-HT7
0460Cinanserin hydrochloride
Selective 5-HT2 antagonist
0462(E)-Capsaicin
Prototypic vanilloid receptor agonist
0463(Z)-Capsaicin
Cis isomer of (E)-Capsaicin (0462)
0464Capsazepine
Vanilloid receptor antagonist. Also activator of ENaCδ
0468N1,N11-Diethylnorspermine tetrahydrochloride
Spermine and spermidine acetyltransferase potentiator
0469Nitrocaramiphen hydrochloride

Muscarinic antagonist, M1 > M2

0471(+)-U-50488 hydrochloride
Less active enantiomer of Cat. No. 0495
0474Dihydroergocristine mesylate

Partial α agonist. Non selective

0475Dihydroergotamine mesylate

Partial α agonist. Non selective

04762,4-Diamino-6-hydroxypyrimidine
Inhibits biosynthesis of tetrahydrobiopterin and thus NOS
0477(±)-Decanoylcarnitine chloride
Intermediate in lipid metabolism
0478Flurofamide
Urease inhibitor
0479Malonoben
Oxidative phosphorylation uncoupler
0481Dilazep dihydrochloride
Adenosine uptake inhibitor
04824-DAMP

Muscarinic M3 antagonist

0483OR-486
Catechol-O-methyl transferase inhibitor
0484Dioctanoylglycol
Diacylglycerol kinase inhibitor
0485Alrestatin
Aldose reductase inhibitor
04861,3-Dipropyl-8-phenylxanthine
A1 selective antagonist
0493AG 18
EGFR/PDGFR-kinase inhibitor
0495(±)-U-50488 hydrochloride
Standard selective κ agonist
0496(-)-U-50488 hydrochloride
More active enantiomer of Cat. No. 0495
0497AG 99
EGFR-kinase inhibitor
0498U-54494A hydrochloride
κ agonist
0500N1,N12-Diethylspermine tetrahydrochloride
Polyamine synthase inhibitor
 
1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 All
[top]