Zolantidine Dimaleate | Histamine Receptors | Potent, Centrally Active H2 Antagonist

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Cat.No.	Product Name
1070	Zolantidine dimaleate

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Zolantidine dimaleate

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Chemical Name: N-[3-[3-(1-Piperidinylmethyl)phenoxy]propyl]-2-benzothi azolamine dimaleate

Biological Activity:

A potent, selective and brain penetrating H₂ receptor antagonist.

Technical Data:

M.Wt:	613.68
Formula:	C₂₂H₂₇N₃OS.2C₄H₄O₄
Storage:	Desiccate at +4°C
Solubility:	Soluble to 100 mM in Water
CAS No:	[104076-38-2]

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References:

Calcutt et al (1988) Zolantidine (SK&F 95282) is a potent selective brain penetrating histamine H₂-receptor antagonist. Br.J.Pharmacol. 93 69. Coruzzi et al (1994) Activity of the new histamine H₂-receptor antagonist zolantidine at cardiac and gastric H₂ receptors. Pharmacology 48 69. Coruzzi et al (1996) Cardiac and gastric effects of histamine H₂ receptor antagonists: no evidence for a correlation between lipophilicity and receptor affinity. Br.J.Pharmacol. 118 1813.

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Keywords: Zolantidine Dimaleate, Histamine Receptors, Potent, Centrally Active H2 Antagonist, Tocris Bioscience

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