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Category:
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7TM Receptors Adrenergic ReceptorsBeta-2 Receptors
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Cat.No.
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Product Name
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1051 |
Zinterol hydrochloride
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| Alternative name(s): |
MJ 9184 |
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Price and Availability
Click here for full price details of
Zinterol
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Chemical Name:
N-[5-[2-[(1,1-Dimethyl-2-phenylethyl)amino]-1-hydroxyet
hyl]-2-hydroxyphenyl]methanesulphonamide hydrochloride |
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Biological Activity:
Potent and selective β2-adrenoceptor agonist
(pKB values are 8.3 and < 5.7 for β2 and β1 receptors respectively,
as measured in human artery).
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
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References:
Kaumann
(1997) Four β-adrenoceptor subtypes in the mammalian heart. TiPS 18 70.
Arvydas Skeberdis et al (1997) Beta-2 adrenergic activation of
L-type Ca2+ current in cardiac myocytes. J.Pharmacol.Exp.Ther. 283
452. Hutchinson et al (2006) Agonist effects of zinterol at the
mouse and human β3-adrenoceptor. Naunyn-Schmied.Arch.Pharmacol. 373 158.
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Keywords: Zinterol, Adrenergic Receptors, Selective B2 Agonist, MJ 9184, Tocris Bioscience
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