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Category:
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7TM Receptors Glutamate (Metabotropic) ReceptorsGroup I mGlu ReceptorsAntagonists
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Cat.No.
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Product Name
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2447 |
Desmethyl-YM 298198
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Price and Availability
Click here for full price details of
Desmethyl-YM 298198
Other Information:
Sold with the permission of Astellas Pharma Inc.
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Chemical Name:
6-Amino-N-cyclohexyl-3-methylthiazolo[3,2-a]benzimidazo
le-2-carboxamide hydrochloride |
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Biological Activity:
Derivative
of the mGlu1-selective antagonist YM 298198 (Cat. No. 2448).
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
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References:
Kohara et al (2005) Radioligand binding properties and pharmacological
characterization of 6-Amino-N-cyclohexyl-N,3-dimethyl-thiazolo[3,2-a]-benzimidazole-2-carboxamide
(YM-298198), a high-affinity, selective and noncompetitive antagonist of
metabotropic glutamate receptor type 1. J.Pharmacol.Exp.Ther. 315 163.
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Keywords: Desmethyl-YM 298198, Glutamate (Metabotropic) Receptors, Derivative Of MGlu1 Antagonist YM 298198, Tocris Bioscience
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