SLIGKV-NH2 | Peptides (Cardiovascular) | PAR2 Receptor Agonist | SLIGKV-amide

Category:

7TM Receptors

Peptides (Cardiovascular)

PAR Receptors

Cat.No.

Product Name

3010

SLIGKV-NH2

Alternative name(s):

SLIGKV-amide

Price and Availability

Click here for full price details of
SLIGKV-NH2

Biological Activity:

Proteinase-activated receptor 2 (PAR2) agonist (K_i = 9.64 μM and IC₅₀ = 10.4 μM). Corresponds to the tethered ligand exposed by trypsin cleavage.

Technical Data:

M.Wt:	614.78
Formula:	_C28H54N8O7
Storage:	Desiccate at -20°C
CAS No:	[190383-13-2]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

References:

Bohm et al (1996) Molecular cloning, expression and potential functions of the human proteinase-activated receptor-2. Biochem.J. 314 1009. Hollenberg and Compton (2002) International union of pharmacology. XXVIII. Proteinase-activated receptors. Pharmacol.Rev. 54 203. Kanke et al (2005) Binding of a highly potent protease-activated receptor-2 (PAR2) activating peptide, [³H]2-furoyl-LIGRL-NH₂, to human PAR2. Br.J.Pharmacol. 145 255.

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Keywords: SLIGKV-NH2, Peptides (Cardiovascular), PAR2 Receptor Agonist, SLIGKV-amide, Tocris Bioscience

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