Ac-RYYRWK-NH2 | Opioid Receptors | Potent, Selective ORL1 Partial Agonist Peptide | AcRYYRWK-NH2

Category:

Cat.No.	Product Name
1387	Ac-RYYRWK-NH₂

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Ac-RYYRWK-NH2

Biological Activity:

Potent, selective partial agonist peptide for the ORL₁ receptor (K_i = 0.71 nM). Selective over μ, δ and κ opioid receptors (IC₅₀ > 4000 nM). Increases food intake in vivo.

Technical Data:

M.Wt:	1012.17
Formula:	C₄₉H₆₉N₁₅O₉
Storage:	Desiccate at -20°C
CAS No:	[200959-47-3]

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References:

Dooley et al (1997) Binding and in vitro activities of peptides with high affinity for the nociceptin/orphanin FQ receptor, ORL₁. J.Pharmacol.Exp.Ther. 283 735. Ho et al (2000) Characterization of the ORL₁ receptor on adrenergic nerve in the rat anococcygeus. Br.J.Pharmacol. 131 349.

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Keywords: Ac-RYYRWK-NH2, Opioid Receptors, Potent, Selective ORL1 Partial Agonist Peptide, AcRYYRWK-NH2, Tocris Bioscience

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Opioid Receptors
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