4-P-PDOT | Melatonin (MT) Receptors | MT2 Antagonist | AH 024 | 4P-PDOT

Category:

7TM Receptors

Melatonin (MT) Receptors

Cat.No.

Product Name

1034

4-P-PDOT

Alternative name(s):

AH 024

4-P-PDOT C19H21NO 4-Phenyl-2-propionamidotetralin

Price and Availability

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4-P-PDOT

Chemical Name: 4-Phenyl-2-propionamidotetralin

Biological Activity:

Melatonin receptor antagonist, >300-fold selective for the MT₂ (vs MT₁) subtype.

Technical Data:

M.Wt:	279.38
Formula:	C₁₉H₂₁NO
Storage:	Store at RT
Solubility:	Soluble to 100 mM in DMSO and to 100 mM in Ethanol
CAS No:	[134865-74-0]

Resources:

Certificate of Analysis / MSDS:

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References:

Dubocovich et al (1995) Melatonin receptors: are there multiple subtypes? TiPS 16 50. Dubocovich et al (1997) Melatonin receptor antagonists that differentiate between the human Mel_1a and Mel_1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina M_L1 presynaptic heteroceptor. Naunyn-Schmied.Arch. Pharmacol. 355 365.

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Keywords: 4-P-PDOT, Melatonin (MT) Receptors, MT2 Antagonist, AH 024, 4P-PDOT, Tocris Bioscience

Literature in this Area

Scientific Reviews

Melatonin Receptors
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