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Category: EnzymesarrowKinasesarrowProtein Kinase A
Cat.No. Product Name
1882 PKA TocrisetTM
Contents:
cAMPS-Rp, triethylammonium salt (Cat. No. 1337)
competitive antagonist of cAMP-induced PKA activation
8-Bromo-cAMP, sodium salt (Cat. No. 1140)
cell-permeable cAMP analogue; PKA activator
Forskolin (Cat. No. 1099)
cell-permeable activator of adenylyl cylcase
KT 5720 (Cat. No. 1288)
potent, selective inhibitor of PKA
NKH 477 (Cat. No. 1603)
water-soluble analogue of forskolin; activator of adenylyl cyclase
Price and Availability

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PKA Tocriset

Biological Activity:

Contains the above products which can be used to modulate PKA signalling. The products are supplied as lyophilised solids or pre-dissolved in 0.5 ml DMSO at various stock concentrations.

Technical Data:

Please see individual product listings for specific technical data.

Click here for further information about Tocriset purity and uses.

Tocriset booklet:

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For specific/earlier batch please select:  

References:

Please see individual product listings for specific references.
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Keywords: PKA Tocriset, Kinases, Selection Of 5 PKA Modulators (Cat. Nos. 1337, 1140, 1099, 1288 & 1603), PKATocriset, Tocris Bioscience

Literature in this Area
Signal Transduction Guide
Signal Transduction Guide : An informative guide for all scientists working in: Cell cycle & apoptosis, Protein kinases & phosphatases, Ion channels, Calcium & lipid signaling, Cyclic nucleotides & G-proteins, Nitric oxide, & Signaling EnzymesA complete listing of signal transduction products available from Tocris, including descriptions on selected tools and unit sizes.
View PDF
Product Feature
Kinase Inhibitors
Key kinase Inhibitors available from Tocris include:
2718   LY 364947
Selective inhibitor of TGF-β RI
2693   PHA 665752
Potent & selective cMET inhibitor
2605   PD 198306
Potent & selective inhibitor of MEK1/2
2539   IKK 16
Selective inhibitor of IKK
View Product Feature
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