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Category: Ion ChannelsarrowLigand-gated Ion ChannelsarrowAcetylcholine (Nicotinic) ReceptorsarrowOther Acetylcholine
Cat.No. Product Name
0750 PG-9 maleate  
Price and Availability

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PG-9 maleate
Chemical Name: Tropanyl 2-(4-bromophenyl)propionate maleate

Biological Activity:

A potent analgesic and nootropic agent. Increases release of acetylcholine.

Technical Data:

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M.Wt: 468.34
Formula: C17H22BrNO2.C4H4O4
Storage: Store at RT
Solubility: Soluble in DMSO

Resources:

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    • Certificate of Analysis / MSDS:

    Certificate of Analysis is currently unavailable on-line. Please contact Customer Service
    Product/Material Safety Data Sheet: View current batch

    References:

    Gualtieri et al (1994) Presynaptic cholinergic modulators as potent cognition enhancers and analgesic drugs. 1. Tropic and 2-phenylpropionic acid esters. J.Med.Chem. 37 1704. Ghelardini et al (1998) Antinociceptive and antiamnesic properties of the presynaptic cholinergic amplifier PG-9. J.Pharmacol.Exp.Ther. 284 806.

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    Keywords: PG-9 Maleate, Ligand-gated Ion Channels, Presynaptic Cholinergic Modulator , PG9 Maleate, Tocris Bioscience
    Literature in this Area
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    Nicotinic ACh Receptors
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    Signal Transduction Guide
    Signal Transduction Guide : An informative guide for all scientists working in: Cell cycle & apoptosis, Protein kinases & phosphatases, Ion channels, Calcium & lipid signaling, Cyclic nucleotides & G-proteins, Nitric oxide, & Signaling EnzymesA complete listing of signal transduction products available from Tocris, including descriptions on selected tools and unit sizes.
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