Octreotide | Peptides (Hypothalamic / Pituitary Hormones) | Sst2, Sst3 & Sst5 Agonist | SMS 201995 | Sandostatin

Category:

7TM Receptors

Peptides (Hypothalamic/Pituitary Hormones)

Somatostatin Receptors

Cat.No.

Product Name

1818

Octreotide

Alternative name(s):	SMS 201995
	Sandostatin

Price and Availability

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Octreotide

Biological Activity:

Peptide agonist for sst₂, sst₃ and sst₅ somatostatin receptors. IC₅₀/K_d values (nM) at cloned human somatostatin receptors are: 290-1140 (sst₁), 0.4-2.1 (sst₂), 4.4-34.5 (sst₃), > 1000 (sst₄), and 5.6-32 (sst₅).

Technical Data:

M.Wt:	1019.24
Formula:	C₄₉H₆₆N₁₀O₁₀S₂
Storage:	Desiccate at -20°C
CAS No:	[79517-01-4]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

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References:

Raynor et al (1993) Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding to linear peptides. Mol.Pharmacol. 43 838. Hoyer et al (1994) Molecular pharmacology of somatostatin receptors. Naunyn-Schmied.Arch.Pharmacol. 350 441. Hannon et al (2002) Drug design at peptide receptors. Somatostatin receptor ligands. J.Mol.Neurosci. 18 15.

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Keywords: Octreotide, Peptides (Hypothalamic / Pituitary Hormones), Sst2, Sst3 & Sst5 Agonist, SMS 201995, Sandostatin, Tocris Bioscience

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Product Feature

Somatostatin Receptors

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