O-1602 | Cannabinoid Receptors | Potent GPR55 Receptor Agonist | O1602

Category:

Cat.No.	Product Name
2797	O-1602

Price and Availability

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O-1602

Chemical Name: 5-Methyl-4-[(1R,6R)-3-methyl-6-(1-cyclohexen-1-yl]-1,3- benzenediol

Biological Activity:

Analogue of cannabidiol that is a potent agonist at the GPR55 cannabinoid receptor (EC₅₀ values are 13, > 30000 and > 30000 nM for GPR55, CB₁ and CB₂ receptors respectively). Induces activation of RhoA, cdc42 and rac1.

Technical Data:

M.Wt:	258.36
Formula:	_C17H22O2
Storage:	Store at -20°C
Solubility:	Soluble in Methyl acetate (supplied in solution (10mg/ml))
Purity:	>98%
CAS No:	[317321-41-8]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

References:

Ryberg et al (2007) The orphan receptor GPR55 is a novel cannabinoid receptor. Br.J.Pharmacol. 152 1092.

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Keywords: O-1602, Cannabinoid Receptors, Potent GPR55 Receptor Agonist, O1602, Tocris Bioscience

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Cannabinoid Receptors
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