Naloxone Hydrochloride | Opioid Receptors | Broad Spectrum Opioid Antagonist

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Cat.No.	Product Name
0599	Naloxone hydrochloride

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Naloxone hydrochloride

Chemical Name: (5a)- 4,5-Epoxy-3,14-dihydro-17-(2-propenyl)morphinan-6-one hydrochloride

Biological Activity:

Opioid antagonist.

Technical Data:

M.Wt:	363.84
Formula:	C₁₉H₂₁NO₄.HCl
Storage:	Store at RT
Solubility:	Soluble to 100 mM in Water
Purity:	>99%
CAS No:	[357-08-4]

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References:

Merck Index 12 6449. Olson et al (1996) Endogenous opiates: 1995 Peptides 17 1421. Spivak et al (1997) Naloxone activation of mu-opioid receptors mutated at a histidine residue lining the opioid cavity. Mol.Pharmacol. 52 983. Pinelli and Trivulzio (1997) Quantitative evaluation of opioid withdrawal signs in rats repeatedly treated with morphine and injected with naloxone, in the absence or presence of the antiabstinence agent clonidine. J.Pharmacol.Toxicol.Methods 38 117.

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Keywords: Naloxone Hydrochloride, Opioid Receptors, Broad Spectrum Opioid Antagonist, Tocris Bioscience

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Opioid Receptors
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