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Category: 7TM Receptorsarrow5-HT Receptorsarrow5-HT1 Receptorsarrow5-HT1A
Cat.No. Product Name
0553 NAN-190 hydrobromide  
Price and Availability

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NAN-190 hydrobromide
Chemical Name: 1-(2-Methoxyphenyl)-4-(4-phthalimidobutyl)piperazine hydrobromide

Biological Activity:

5-HT1A antagonist.

Technical Data:

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M.Wt: 474.4
Formula: C23H27N3O3.HBr
Storage: Store at RT
Solubility: Soluble to 10 mM in Ethanol
CAS No: [115388-32-4]

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    • Certificate of Analysis / MSDS:

    Certificate of Analysis: View current batch
    Product/Material Safety Data Sheet: View current batch

    References:

    Williams and Glennon (1988) NAN-190: an arylpiperazine analog that antagonizes the stimulus effects of the 5-HT1A agonist 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT). Eur.J.Pharmacol. 154 339. Glennon et al (1988) Arylpiperazine derivatives as high affinity 5-HT1A serotonin ligands.  J.Med.Chem. 31 1968. Dourish (1992) Effects of the putative 5-HT1A receptor antagonist NAN-190 on free feeding and on feeding induced by the 5-HT1A receptor agonist 8-OH-DPAT in the rat. Eur.J.Pharmacol. 219 105.
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    Keywords: NAN-190 Hydrobromide, 5-HT Receptors, 5-HT1A Antagonist, NAN190 Hydrobromide, Tocris Bioscience
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