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Category: 7TM Receptorsarrow5-HT ReceptorsarrowSerotonergic-Related
Cat.No. Product Name
1064 Methysergide maleate
Price and Availability

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Methysergide maleate
Chemical Name: [8b(S)]-9,10-Didehydro-N-[1-(hydroxymethyl)propyl]-1,6- dimethylergoline-8-carboxamide maleate

Biological Activity:

Mixed 5-HT1/5-HT2 receptor antagonist.

Technical Data:

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M.Wt: 469.54
Formula: C21H27N3O2.C4H4O4
Storage: Store at RT
Solubility: Soluble to 10 mM in Water
Purity: >99%
CAS No: [129-49-7]

Resources:

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    References:

    Merck Index 12 6217. Hoyer et al (1994) VII. International Union of Pharmacology classification of receptors for 5-hydroxytryptamine (serotonin). Pharmacol.Rev. 46 157.
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    Keywords: Methysergide Maleate, 5-HT Receptors, 5-HT1 / 5-HT2 Antagonist, Tocris Bioscience

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