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Category: Ion ChannelsarrowLigand-gated Ion Channelsarrow5-HT3 ReceptorsarrowAgonists
Cat.No. Product Name
0566 N-Methylquipazine dimaleate  
Price and Availability

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N-Methylquipazine dimaleate
Chemical Name: 2-(1-N-Methylpiperazinyl)quinoline dimaleate

Biological Activity:

5-HT3 agonist. Has almost the same affinity for 5-HT3 sites as quipazine but unlike the latter, does not bind to 5-HT1B sites.

Technical Data:

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M.Wt: 459.45
Formula: C14H17N3.(C4H4O4)2
Storage: Store at RT
Solubility: Soluble to 50 mM in Water
CAS No: [28614-26-8]

Resources:

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    • Certificate of Analysis / MSDS:

    Certificate of Analysis: View current batch
    Product/Material Safety Data Sheet: View current batch

    References:

    Glennon et al (1989) Binding of arylpiperazines to 5-HT3 serotonin receptors: results of a structure-affinity study. Eur.J.Pharmacol. 168 387.
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    Keywords: N-Methylquipazine Dimaleate, Ligand-gated Ion Channels, 5-HT3 Agonist, NMethylquipazine Dimaleate, Tocris Bioscience
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