Methylergometrine Maleate | 5-HT Receptors | Active Metabolite Of Methysergide | Methylergonovine Maleate

Category:

7TM Receptors

5-HT Receptors

Serotonergic-Related

Cat.No.

Product Name

0549

Methylergometrine maleate

Alternative name(s):

Methylergonovine maleate

Methylergometrine maleate
C20H25N3O2.C4H4O4 [8b(S)]-9,10-Didehydro-N-[1-(hydroxymethyl)propyl]-6-methylergoline-8-carboxamide maleate

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Methylergometrine maleate

Chemical Name: [8b(S)]-9,10-Didehydro-N-[1-(hydroxymethyl)propyl]-6-me thylergoline-8-carboxamide maleate

Biological Activity:

Active metabolite of methysergide; uterotonic agent and oxytocic.

Technical Data:

M.Wt:	455.51
Formula:	C₂₀H₂₅N₃O₂.C₄H₄O₄
Storage:	Desiccate at RT
Solubility:	Soluble to 25 mM in Water
CAS No:	[113-42-8]

Resources:

Certificate of Analysis / MSDS:

Certificate of Analysis: View current batch

Product/Material Safety Data Sheet: View current batch

References:

Merck 12 6147. Muller-Schweinitzer and Tapparelli (1986) Methylergometrine, an active metabolite of methysergide. Cephalalgia 6 35. MacLennan and Martin (1990) Actions of non-peptide ergot alkaloids at 5-HT1-like and 5-HT2 receptors mediating vascular smooth muscle contraction. Naunyn-Schmied.Arch.Pharmacol. 342 120. Pertz (1993) 5-Hydroxytryptamine (5-HT) contracts the guinea-pig isolated iliac artery via 5-HT1-like and 5-HT2 receptors. Naunyn-Schmied.Arch.Pharmacol. 348 558.

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Keywords: Methylergometrine Maleate, 5-HT Receptors, Active Metabolite Of Methysergide, Methylergonovine Maleate, Tocris Bioscience

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