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Category:
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7TM Receptors Adrenergic ReceptorsAlpha-1 ReceptorsOther
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Cat.No.
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Product Name
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0581 |
3-[2-[4-(2-Methoxyphenyl)piperazin-1-yl] ethyl]pyrimido[5,4-b] indole-2,4-dione
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Price and Availability
Click here for full price details of
3-[2-[4-(2-Methoxyphenyl)piperazin-1-yl] ethyl]pyrimido[5,4-b] indole-2,4-dione
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Biological Activity:
Very potent ligand for α1 sites (Ki for displacement of prazosin =
0.2 nM). Also binds to 5-HT1A sites (Ki = 50 nM).
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Technical Data:
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Resources:
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Certificate of Analysis / MSDS:
Certificate of Analysis is currently unavailable on-line. Please contact Customer Service
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References:
Russo et al (1991) Pyrimido[5,4-b]indole derivatives. 1. A new class of potent
and selective α1 adrenoceptor ligands. J.Med.Chem. 34
1850.
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Keywords: 3-[2-[4-(2-Methoxyphenyl)piperazin-1-yl] Ethyl]pyrimido[5,4-b] Indole-2,4-dione, Adrenergic Receptors, A1 Ligand , 3[2-[4-(2-Methoxyphenyl)piperazin-1-yl] Ethyl]pyrimido[5,4-b] Indole-2,4-dione, Tocris Bioscience
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